SCHEMBL7529065

SCHEMBL7529065

O=C1O[C@@H](CN2CCC(Cc3ccccc3)CC2)CN1c1ccc(Cl)cc1

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 4/20 0.57
SLC6A2 P23975 2/20 0.55
SLC6A4 P31645 2/20 0.55
ALDH1A1 P00352 1/20 0.54
SIGMAR1 Q99720 9/20 0.52
HTR1A P08908 4/20 0.52
TMEM97 Q5BJF2 1/20 0.47
CCR3 P51677 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9677253 1.00 GRM2 (0.57) GRM2SLC6A2SLC6A4ALDH1A1SIGMAR1
SCHEMBL9678366 0.92 GRM2 (0.67) GRM2SLC6A2SLC6A4SIGMAR1HTR1A
SCHEMBL7487787 0.90 SIGMAR1 (0.50) GRM2SLC6A2SLC6A4ALDH1A1SIGMAR1
SCHEMBL9844385 0.89 SLC6A2 (0.58) GRM2SLC6A2SLC6A4ALDH1A1CCR3
SCHEMBL9676204 0.89 GRM2 (0.57) GRM2ALDH1A1SIGMAR1HTR1A
SCHEMBL9677541 0.89 GRM2 (0.57) GRM2SIGMAR1HTR1ATMEM97
SCHEMBL9677266 0.89 GRM2 (0.54) GRM2SLC6A2SLC6A4ALDH1A1SIGMAR1
Hydrochloric Acid SCHEMBL9679291 0.88 GRM2 (0.56) GRM2ALDH1A1SIGMAR1HTR1A
SCHEMBL9678853 0.86 SIGMAR1 (0.65) GRM2SIGMAR1
SCHEMBL7481896 0.86 GRM2 (0.58) GRM2SIGMAR1HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002030422-A1 USE OF DEFINED SUBSTANCES THAT BIND TO THE SIGMA RECEPTOR FOR COMBATING SARCOMA AND CARCINOMA MERCK PATENT GMBH (DE) 2002-04-18 WO claimed
WO-2002030422-A1 USE OF DEFINED SUBSTANCES THAT BIND TO THE SIGMA RECEPTOR FOR COMBATING SARCOMA AND CARCINOMA MERCK PATENT GMBH (DE) 2002-04-18 WO disclosed
WO-2002030422-A1 USE OF DEFINED SUBSTANCES THAT BIND TO THE SIGMA RECEPTOR FOR COMBATING SARCOMA AND CARCINOMA MERCK PATENT GMBH (DE) 2002-04-18 WO disclosed