SCHEMBL7529482

SCHEMBL7529482

CC(=O)NC(C(=O)NCc1ccccc1F)c1ccoc1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC1A2 P43004 1/20 0.45
HPGD P15428 3/20 0.44
ALDH1A1 P00352 3/20 0.44
MAPT P10636 1/20 0.44
TSHR P16473 1/20 0.44
RIPK1 Q13546 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.39
HIF1A Q16665 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C19 P33261 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
FOLH1 Q04609 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7526519 0.83 CA12 (0.52) HPGDALDH1A1TSHRSMN1; SMN2CYP3A4
SCHEMBL1710160 0.81 HPGD (0.48) SLC1A2HPGDALDH1A1MAPTTSHR
SCHEMBL9137159 0.81 HPGD (0.43) HPGDALDH1A1TSHR
SCHEMBL7528147 0.80 ANPEP (0.46) HPGDALDH1A1CYP2C19FOLH1
SCHEMBL2905073 0.72 SLC1A2 (0.65) SLC1A2HPGDALDH1A1MAPTTSHR
SCHEMBL1685923 0.72 RIPK1 (0.61) SLC1A2HPGDALDH1A1MAPTTSHR
SCHEMBL29941696 0.72 RIPK1 (0.61) SLC1A2HPGDALDH1A1MAPTTSHR
SCHEMBL7521866 0.69 CCR2 (0.43) HPGDALDH1A1MAPTTSHR
SCHEMBL25259336 0.69 SLC1A2 (0.60) SLC1A2HPGDALDH1A1MAPTTSHR
SCHEMBL25209028 0.69 SLC1A2 (0.60) SLC1A2HPGDALDH1A1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0400440-B1 Amino acid derivative anticonvulsant RES CORP TECHNOLOGIES INC (US) 2002-03-13 EP disclosed
US-5654301-A Lacosamide FDA Orange book listed patent RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1997-08-05 US disclosed
US-5378729-A Diamide derivatives RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1995-01-03 US disclosed
WO-1992021648-A1 AMINO ACID DERIVATIVE ANTICONVULSANT RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1992-12-10 WO disclosed
WO-1990015069-A2 AMINO ACID DERIVATIVE ANTICONVULSANT RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1990-12-13 WO disclosed
EP-0400440-A1 Amino acid derivative anticonvulsant RESEARCH CORPORATION TECHNOLOGIES, INC. (US) 1990-12-05 EP disclosed