SCHEMBL7529762

SCHEMBL7529762

COc1ccc(N=C=O)c(OC)c1.COc1ccccc1N=C=O

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.61
CYP3A4 P08684 4/20 0.61
HPGD P15428 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
CYP1B1 Q16678 6/20 0.44
CYP1A1 P04798 5/20 0.44
CYP1A2 P05177 5/20 0.44
MAPT P10636 5/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KMT2A Q03164 2/20 0.43
NPC1 O15118 1/20 0.43
PKM P14618 1/20 0.43
RAB9A P51151 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
GAA P10253 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29541267 0.92 ALDH1A1 (0.71) ALDH1A1CYP3A4HPGDTDP1CYP1B1
SCHEMBL703276 0.92 ALDH1A1 (0.71) ALDH1A1CYP3A4HPGDTDP1CYP1B1
SCHEMBL77114 0.87 ALDH1A1 (0.61) ALDH1A1CYP3A4HPGDTDP1MAPT
SCHEMBL29471398 0.87 ALDH1A1 (0.61) ALDH1A1CYP3A4HPGDTDP1MAPT
SCHEMBL8943270 0.85 CYP3A4 (0.50) ALDH1A1CYP3A4HPGDTDP1CYP1A2
SCHEMBL8942826 0.84 ALDH1A1 (0.61) ALDH1A1CYP3A4HPGDTDP1CYP1B1
SCHEMBL11194657 0.83 ALDH1A1 (0.69) ALDH1A1CYP3A4HPGDTDP1CYP1B1
SCHEMBL374346 0.82 ALDH1A1 (0.56) ALDH1A1CYP3A4HPGDTDP1CYP1B1
SCHEMBL29538723 0.82 ALDH1A1 (0.56) ALDH1A1CYP3A4HPGDTDP1CYP1B1
SCHEMBL14895167 0.79 CYP3A4 (0.77) ALDH1A1CYP3A4HPGDTDP1CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP disclosed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO disclosed