SCHEMBL7530474

SCHEMBL7530474

O=C(O)CCCOc1cc([N+](=O)[O-])ccc1CO

nearest known ligand 0.49

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.47
CYSLTR2 Q9NS75 1/20 0.47
CYSLTR1 Q9Y271 1/20 0.47
TSHR P16473 2/20 0.46
TDP1 Q9NUW8 2/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.46
MAPT P10636 4/20 0.46
ALDH1A1 P00352 3/20 0.46
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
CYP19A1 P11511 3/20 0.46
CYP11B1 P15538 3/20 0.46
CYP11B2 P19099 3/20 0.46
RAB9A P51151 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.43
POLB P06746 1/20 0.43
LTB4R Q15722 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14035613 0.83 ALDH1A1 (0.53) CYP1A2CYSLTR2CYSLTR1TSHRTDP1
SCHEMBL25412691 0.82 MAPT (0.50) CYP1A2CYSLTR2CYSLTR1TSHRTDP1
SCHEMBL31534614 0.82 RAB9A (0.55) CYP1A2CYSLTR2CYSLTR1TSHRTDP1
SCHEMBL7521060 0.81 TDP1 (0.51) CYP1A2TSHRTDP1MAPTALDH1A1
SCHEMBL7519738 0.80 CHRNB2 (0.48) CYP1A2TSHRTDP1MAPTALDH1A1
SCHEMBL12190689 0.79 MAPT (0.49) CYP1A2TSHRTDP1MAPTALDH1A1
SCHEMBL14008900 0.77 CYP19A1 (0.62) MAPTALDH1A1MEN1KMT2ACYP19A1
SCHEMBL8163799 0.76 MAPT (0.66) CYP1A2TSHRTDP1MAPTALDH1A1
SCHEMBL8159350 0.76 MAPT (0.55) CYSLTR2CYSLTR1TSHRTDP1PTGDR2
SCHEMBL27837027 0.76 CYSLTR2 (0.55) CYP1A2CYSLTR2CYSLTR1MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173414-A1 N-PROTECTED AMINES AND THEIR USE AS PRODRUGS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2002-01-23 EP disclosed
WO-2000064864-A9 N-PROTECTED AMINES AND THEIR USE AS PRODRUGS CANCER RES CAMPAIGN TECH (GB) 2001-12-27 WO disclosed
WO-2000064864-A1 N-PROTECTED AMINES AND THEIR USE AS PRODRUGS CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2000-11-02 WO disclosed