SCHEMBL7530816

SCHEMBL7530816

Cc1ncc(-c2ccsc2C(N)=O)s1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.47
GRM2 Q14416 3/20 0.39
NR1I2 O75469 1/20 0.39
LIMK1 P53667 2/20 0.38
HCAR2 Q8TDS4 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37
PIK3CD O00329 2/20 0.37
PLA2G10 O15496 1/20 0.37
IKBKB O14920 3/20 0.36
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 2/20 0.36
POLB P06746 1/20 0.36
HTT P42858 1/20 0.36
CDK8 P49336 1/20 0.36
CDK19 Q9BWU1 1/20 0.36
EDNRA P25101 1/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36
PIK3C3 Q8NEB9 1/20 0.36
PKM P14618 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31661900 0.74 BCAT2 (0.57) BCAT2LIMK1PLA2G10IKBKBKDM4E
SCHEMBL1685092 0.74 PIK3CD (0.54) BCAT2GRM2NR1I2HCAR2PIK3CD
SCHEMBL31661857 0.70 SIRT3 (0.50) BCAT2LIMK1CDK8
SCHEMBL31661830 0.70 MKNK1 (0.54) BCAT2LIMK1PLA2G10IKBKBKDM4E
SCHEMBL16011605 0.69 BCAT2 (0.59) BCAT2LIMK1IKBKBKDM4EALDH1A1
SCHEMBL2231308 0.69 BCAT2 (0.69) BCAT2GRM2PLA2G10IKBKBKDM4E
SCHEMBL31661820 0.69 BCAT2 (0.58) BCAT2LIMK1KDM4EALDH1A1POLB
SCHEMBL12495840 0.68 BCAT2 (0.62) BCAT2IKBKBKDM4EALDH1A1POLB
SCHEMBL27711486 0.68 BCAT2 (0.49) BCAT2LIMK1PLA2G10IKBKBKDM4E
SCHEMBL27596977 0.68 PIK3CD (0.40) GRM2NR1I2HCAR2NPSR1PIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002017358-A2 QUINUCLIDINE-SUBSTITUTED HETEROARYL MOIETIES FOR TREATMENT OF DISEASE (NICOTINIC ACETYLCHOLINE RECEPTOR ANTAGONISTS) PHARMACIA & UPJOHN COMPANY (US) 2002-02-28 WO claimed