SCHEMBL7530892

SCHEMBL7530892

COc1cc2c(cc1C=O)C(C)(C(F)(F)F)OC2=O

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.41
KDM4E B2RXH2 2/20 0.41
TSHR P16473 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.38
GAA P10253 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
SIRT1 Q96EB6 1/20 0.34
ACHE P22303 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MAPT P10636 1/20 0.33
PRKDC P78527 1/20 0.33
ERN1 O75460 5/20 0.32
KMT2A Q03164 1/20 0.32
TLR2 O60603 1/20 0.31
TLR1 Q15399 1/20 0.31
TLR6 Q9Y2C9 1/20 0.31
FGFR1 P11362 1/20 0.31
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7532238 0.79 SIRT1 (0.40) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL6402101 0.74 ALDH1A1 (0.42) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL7247609 0.74 ALDH1A1 (0.42) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL7535419 0.72 PDK2 (0.50) ALDH1A1KDM4ETDP1
SCHEMBL7537870 0.72 PDK2 (0.50) ALDH1A1KDM4ETDP1
SCHEMBL7539368 0.72 PDK2 (0.50) ALDH1A1KDM4ETDP1
SCHEMBL6406585 0.72 TACR1 (0.44) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL6400790 0.72 TACR1 (0.44) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL6400684 0.72 TACR1 (0.44) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL6401662 0.67 ALDH1A1 (0.43) ALDH1A1KDM4ETSHRTDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032571-B1 PIPERIDINYLAMINOMETHYL TRIFLUOROMETHYL CYCLIC ETHER COMPOUNDS AS SUBSTANCE P ANTAGONISTS PFIZER (US) 2002-06-12 EP claimed