SCHEMBL7532238

SCHEMBL7532238

COc1cc2c(cc1C=O)C(c1ccccc1)(C(F)(F)F)OC2=O

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SIRT1 Q96EB6 3/20 0.40
TP53 P04637 1/20 0.37
ALDH1A1 P00352 5/20 0.37
KDM4E B2RXH2 1/20 0.37
TSHR P16473 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
FGFR1 P11362 1/20 0.35
LMNA P02545 1/20 0.35
HPGD P15428 1/20 0.35
MDM2 Q00987 1/20 0.34
ERN1 O75460 4/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
MAPT P10636 1/20 0.33
NPC1 O15118 2/20 0.33
POLB P06746 1/20 0.33
RAB9A P51151 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7530892 0.79 ALDH1A1 (0.41) SIRT1ALDH1A1KDM4ETSHRTDP1
SCHEMBL6400844 0.78 ALDH1A1 (0.38) SIRT1ALDH1A1KDM4ETSHRTDP1
SCHEMBL7537292 0.77 TP53 (0.51) SIRT1TP53ALDH1A1KDM4ETDP1
SCHEMBL5083219 0.65 AVPR1A (0.40) SIRT1TP53ALDH1A1KDM4ESMN1; SMN2
SCHEMBL9717769 0.65 ALDH1A1 (0.58) ALDH1A1KDM4ETSHRTDP1FGFR1
SCHEMBL6401662 0.63 ALDH1A1 (0.43) ALDH1A1KDM4ETSHRTDP1LMNA
SCHEMBL6224414 0.62 ALDH1A1 (0.58) ALDH1A1KDM4ETSHRTDP1FGFR1
SCHEMBL918824 0.62 CYP1A1 (0.61) ALDH1A1KDM4ETSHRTDP1FGFR1
SCHEMBL918825 0.62 CYP1A1 (0.61) ALDH1A1KDM4ETSHRTDP1FGFR1
SCHEMBL19662549 0.62 GPR35 (0.41) TP53ALDH1A1KDM4ETDP1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1032571-B1 PIPERIDINYLAMINOMETHYL TRIFLUOROMETHYL CYCLIC ETHER COMPOUNDS AS SUBSTANCE P ANTAGONISTS PFIZER (US) 2002-06-12 EP claimed