SCHEMBL7533909

SCHEMBL7533909

CCCc1ccccc1NC=O

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
TSHR P16473 1/20 0.41
ALDH1A1 P00352 2/20 0.39
TLR8 Q9NR97 1/20 0.37
PABPC1 P11940 1/20 0.36
POLB P06746 1/20 0.36
P2RX7 Q99572 1/20 0.35
GAA P10253 2/20 0.35
MAPT P10636 1/20 0.35
TAS1R3 Q7RTX0 1/20 0.35
TAS1R1 Q7RTX1 1/20 0.35
SCD O00767 1/20 0.34
CLCN2 P51788 1/20 0.33
CTSL P07711 1/20 0.33
CTSS P25774 1/20 0.33
CTSK P43235 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14390806 0.89 CYP3A4 (0.44) TSHRALDH1A1TLR8POLBSCD
SCHEMBL21995029 0.88 TSHR (0.46) TSHRALDH1A1PABPC1GAAMAPT
SCHEMBL5536492 0.86 LIPG (0.49) MAPT
SCHEMBL1685968 0.86 LIPG (0.49) MAPT
SCHEMBL33525287 0.86 ALDH1A1 (0.46) TSHRALDH1A1POLBGAAMAPT
SCHEMBL2243716 0.86 ALDH1A1 (0.46) TSHRALDH1A1POLBGAAMAPT
SCHEMBL26456221 0.81 TAAR1 (0.46) TSHRALDH1A1GAAMAPT
SCHEMBL5219876 0.81 TSHR (0.41) TSHRALDH1A1PABPC1
SCHEMBL12569376 0.81 TAAR1 (0.45) ADRA2CTSHRALDH1A1PABPC1CTSK
SCHEMBL12571394 0.81 TAAR1 (0.45) ADRA2CTSHRALDH1A1PABPC1CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP claimed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US claimed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO claimed
EP-2847193-B1 HETEROARYL COMPOUNDS AND METHODS OF USE THEREOF SUNOVION PHARMACEUTICALS INC (US) 2019-08-07 EP disclosed
EP-1770086-A1 Selected CGRP antagonists, process for their preparation as well as their use as medicaments Boehringer Ingelheim Pharma GmbH & Co. KG (DE) 2007-04-04 EP disclosed
EP-1189891-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION Bioscience AG (DE) 2002-03-27 EP disclosed
US-6362342-B1 BIOSYNTHESIS; DRUG LIBRARIES LION BIOSCIENCE AG (DE) 2002-03-26 US disclosed
WO-2001000594-A1 TRIAZOLE COMPOUNDS AND COMBINATORIAL LIBRARIES THEREOF LION BIOSCIENCE AG (DE) 2001-01-04 WO disclosed