SCHEMBL7534135

SCHEMBL7534135

CC(C)COc1cc(C(C)N(C)C)ccc1-c1cccc(N)n1

nearest known ligand 0.45

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 16/20 0.45
NOS3 P29474 12/20 0.44
NOS2 P35228 8/20 0.44
TLR8 Q9NR97 1/20 0.39
CHRNA7 P36544 1/20 0.38
MCHR1 Q99705 1/20 0.37
IDH1 O75874 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7534301 0.79 NOS1 (0.47) NOS1NOS3NOS2MCHR1
SCHEMBL6700027 0.73 NOS1 (0.50) NOS1NOS3NOS2
SCHEMBL6700692 0.71 NOS1 (0.52) NOS1NOS3NOS2
SCHEMBL27517402 0.71 NOS3 (0.39) NOS1NOS3NOS2
SCHEMBL6698874 0.70 NOS1 (0.43) NOS1NOS3NOS2MCHR1
SCHEMBL6700030 0.70 NOS1 (0.58) NOS1NOS3NOS2
SCHEMBL218971 0.67 MCHR1 (0.45) NOS1NOS3NOS2TLR8MCHR1
SCHEMBL220790 0.66 NOS1 (0.58) NOS1NOS3NOS2
SCHEMBL221742 0.66 NOS1 (0.51) NOS1NOS3NOS2TLR8MCHR1
SCHEMBL21223572 0.65 TLR8 (0.50) TLR8CHRNA7MCHR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1007512-B1 BRANCHED ALKOXY-SUBSITUTED 2-AMINOPYRIDINES AS NOS INHIBITORS PFIZER PROD INC (US) 2002-04-03 EP claimed