SCHEMBL7534601

SCHEMBL7534601

CCOc1c(N)cccc1C(N)=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.49
HSD17B10 Q99714 4/20 0.49
TSHR P16473 2/20 0.45
PARP10 Q53GL7 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
LMNA P02545 2/20 0.43
NR1I2 O75469 1/20 0.43
CHRM2 P08172 1/20 0.43
CYP3A4 P08684 1/20 0.43
ADRA2A P08913 1/20 0.43
MAPT P10636 1/20 0.43
OPRK1 P41145 1/20 0.43
HTR2B P41595 1/20 0.43
SLC6A3 Q01959 1/20 0.43
HDAC6 Q9UBN7 1/20 0.43
KDM4E B2RXH2 1/20 0.43
PKM P14618 1/20 0.43
CFTR P13569 1/20 0.41
PARP1 P09874 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2923268 0.86 MMP2 (0.50) ALDH1A1HSD17B10TSHRMEN1KMT2A
SCHEMBL28189538 0.83 ALDH1A1 (0.59) ALDH1A1HSD17B10TSHRKMT2ALMNA
SCHEMBL28309500 0.83 L3MBTL1 (0.45) ALDH1A1HSD17B10TSHRPARP10MEN1
SCHEMBL288797 0.83 TSHR (0.45) ALDH1A1HSD17B10TSHRPARP10MEN1
SCHEMBL3189724 0.83 TSHR (0.53) TSHRMEN1KMT2ALMNANR1I2
SCHEMBL15713724 0.83 KDM4E (0.40) ALDH1A1HSD17B10TSHRMEN1KMT2A
SCHEMBL3476584 0.81 PARP10 (0.46) ALDH1A1HSD17B10TSHRPARP10MEN1
SCHEMBL31314603 0.81 TSHR (0.44) ALDH1A1TSHRPARP10MEN1KMT2A
SCHEMBL29686816 0.81 TSHR (0.53) ALDH1A1TSHRPARP10MEN1KMT2A
SCHEMBL28706339 0.81 TSHR (0.53) ALDH1A1TSHRPARP10MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102391222-B As the hydroxamic acid ester of therapeutical agent PHARMACYCLICS INC. (US) 2015-10-21 CN disclosed
EP-1196404-A1 PIPERAZINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Astrazeneca UK Limited (GB) 2002-04-17 EP disclosed
WO-2001002381-A1 PIPERAZINE DERIVATIVES AS MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY ASTRAZENECA UK LIMITED (GB) 2001-01-11 WO disclosed