SCHEMBL7535919

SCHEMBL7535919

CN(C)c1cccc(CN2CC=C(c3c[nH]c4ccc(Cl)cc34)CC2)c1

nearest known ligand 0.76

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.76
OPRK1 P41145 1/20 0.76
DRD2 P14416 17/20 0.62
HTR1A P08908 16/20 0.62
HTR2A P28223 3/20 0.59
HTT P42858 1/20 0.59
SLC6A4 P31645 5/20 0.57
HTR6 P50406 5/20 0.54
HTR7 P34969 4/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14280720 0.87 OPRM1 (1.00) OPRM1OPRK1DRD2HTR1AHTR2A
Hydrochloric Acid SCHEMBL11320856 0.79 OPRM1 (0.73) OPRM1OPRK1DRD2HTR1ASLC6A4
SCHEMBL11327571 0.79 OPRM1 (0.73) OPRM1OPRK1DRD2HTR1ASLC6A4
SCHEMBL7647977 0.78 SLC6A4 (0.55) OPRM1OPRK1DRD2HTR1ASLC6A4
Tepirindole SCHEMBL11307437 0.78 SLC6A4 (0.72) OPRM1OPRK1DRD2HTR1ASLC6A4
Tepirindole SCHEMBL635174 0.78 SLC6A4 (0.72) OPRM1OPRK1DRD2HTR1ASLC6A4
Tepirindole SCHEMBL29710897 0.78 SLC6A4 (0.72) OPRM1OPRK1DRD2HTR1ASLC6A4
SCHEMBL7536094 0.76 OPRM1 (0.78) OPRM1OPRK1DRD2HTR1AHTR2A
SCHEMBL9527241 0.76 OPRM1 (0.78) OPRM1OPRK1DRD2HTR1AHTR2A
SCHEMBL10366941 0.75 OPRM1 (0.71) OPRM1OPRK1DRD2HTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6476028-B1 Compounds and methods SMITHKLINE BEECHAM CORPORATION 2002-11-05 US claimed
EP-1037635-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2002-11-13 EP disclosed
US-6476028-B1 Compounds and methods SMITHKLINE BEECHAM CORPORATION 2002-11-05 US disclosed
EP-1037635-A1 COMPOUNDS AND METHODS Smithkline Beecham (US) 2000-09-27 EP disclosed
WO-1999017773-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-04-15 WO disclosed