SCHEMBL7536094

SCHEMBL7536094

Oc1ccc2[nH]cc(C3=CCN(Cc4ccccc4)CC3)c2c1

nearest known ligand 0.78

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.78
OPRK1 P41145 1/20 0.78
HTR1A P08908 15/20 0.75
DRD2 P14416 15/20 0.75
HTR2A P28223 5/20 0.75
HTT P42858 1/20 0.75
CYP1A2 P05177 1/20 0.57
CYP3A4 P08684 1/20 0.57
MAPT P10636 1/20 0.57
CYP2C9 P11712 1/20 0.57
TSHR P16473 1/20 0.57
DRD4 P21917 1/20 0.57
CYP2C19 P33261 1/20 0.57
DRD3 P35462 1/20 0.57
TDP1 Q9NUW8 1/20 0.57
KDM4E B2RXH2 1/20 0.55
LMNA P02545 1/20 0.55
ALOX15 P16050 1/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14280720 0.88 OPRM1 (1.00) OPRM1OPRK1HTR1ADRD2HTR2A
SCHEMBL9527241 0.87 OPRM1 (0.78) OPRM1OPRK1HTR1ADRD2HTR2A
SCHEMBL7543848 0.86 HTR1A (1.00) OPRM1OPRK1HTR1ADRD2HTR2A
SCHEMBL7649906 0.85 HTR1A (0.83) OPRM1OPRK1HTR1ADRD2HTR2A
SCHEMBL7859795 0.84 OPRM1 (0.74) OPRM1OPRK1HTR1ADRD2HTR2A
SCHEMBL4194997 0.84 HTR1A (1.00) OPRM1OPRK1HTR1ADRD2HTR2A
SCHEMBL1122147 0.82 OPRM1 (0.71) OPRM1OPRK1HTR1ADRD2HTR2A
Fumaric Acid SCHEMBL9764481 0.80 OPRM1 (0.65) OPRM1OPRK1HTR1ADRD2HTR2A
SCHEMBL8914068 0.80 OPRM1 (0.65) OPRM1OPRK1HTR1ADRD2HTR2A
Maleic Acid SCHEMBL9764477 0.80 OPRM1 (0.65) OPRM1OPRK1HTR1ADRD2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6476028-B1 Compounds and methods SMITHKLINE BEECHAM CORPORATION 2002-11-05 US claimed
EP-1037635-A4 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORP (US) 2002-11-13 EP disclosed
US-6476028-B1 Compounds and methods SMITHKLINE BEECHAM CORPORATION 2002-11-05 US disclosed
EP-1037635-A1 COMPOUNDS AND METHODS Smithkline Beecham (US) 2000-09-27 EP disclosed
WO-1999017773-A1 COMPOUNDS AND METHODS SMITHKLINE BEECHAM CORPORATION (US) 1999-04-15 WO disclosed