SCHEMBL7539758

SCHEMBL7539758

NCc1ccc(-c2noc(=O)[nH]2)nc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
KMO O15229 1/20 0.40
PLA2G2A P14555 7/20 0.36
TRPM8 Q7Z2W7 1/20 0.35
CYP4F2 P78329 1/20 0.34
CYP4A11 Q02928 1/20 0.34
RARB P10826 1/20 0.33
PDE10A Q9Y233 2/20 0.33
ADH5 P11766 1/20 0.33
HIF1A Q16665 1/20 0.33
CTNNB1 P35222 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16285371 0.85 ALDH1A1 (0.48) ALDH1A1KMOPLA2G2ATRPM8RARB
SCHEMBL5009740 0.78 LOXL2 (0.46) ALDH1A1KMOADH5
Hydrochloric Acid SCHEMBL1272214 0.76 ALDH1A1 (0.55) ALDH1A1PLA2G2ARARBADH5
SCHEMBL16285376 0.76 CCR1 (0.48) ALDH1A1KMOPLA2G2ARARBADH5
SCHEMBL21676846 0.73 KMO (0.39) ALDH1A1KMOPLA2G2ATRPM8HIF1A
SCHEMBL31546321 0.73 ALDH1A1 (0.51) ALDH1A1KMOPLA2G2ACYP4F2CYP4A11
SCHEMBL21676847 0.73 MRGPRX4 (0.44) KMO
SCHEMBL351473 0.72 LOXL2 (0.46)
SCHEMBL9771736 0.69 BTK (0.54) ALDH1A1KMOHIF1A
SCHEMBL1098065 0.67 KMO (0.43) ALDH1A1KMOPLA2G2ARARBADH5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1169318-A1 PRODRUGS OF THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2002-01-09 EP disclosed
WO-2000061577-A1 PRODRUGS OF THROMBIN INHIBITORS BASF AKTIENGESELLSCHAFT (DE) 2000-10-19 WO disclosed