SCHEMBL7540320

SCHEMBL7540320

Cc1cccc2[nH]c(C(=O)N[C@H](C(=O)NC(CC(=O)O)C(=O)COc3ccccc3F)C(C)C)c(CC(C)C)c12

nearest known ligand 0.49

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 20/20 0.49
CASP6 P55212 17/20 0.45
CASP8 Q14790 17/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7535127 0.90 CASP3 (0.47) CASP3CASP6CASP8
SCHEMBL7538962 0.89 CASP3 (0.58) CASP3CASP6CASP8
SCHEMBL8606968 0.86 CASP3 (0.41) CASP3CASP6CASP8
SCHEMBL7535627 0.84 CASP3 (0.40) CASP3CASP6CASP8
SCHEMBL7543444 0.81 CASP3 (0.49) CASP3CASP6CASP8
SCHEMBL8608833 0.77 CASP3 (0.44) CASP3CASP6CASP8
SCHEMBL7536449 0.76 MMP2 (0.36) CASP3CASP6CASP8
SCHEMBL27583485 0.76 CASP3 (0.53) CASP3CASP6CASP8
SCHEMBL7201348 0.76 CASP3 (0.53) CASP3CASP6CASP8
SCHEMBL5970017 0.75 CASP3 (0.42) CASP3CASP6CASP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1159291-A1 C-TERMINAL MODIFIED (N-SUBSTITUTED)-2-INDOLYLCARBONYLDIPEPTIDES AS INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES Idun Pharmaceuticals, Inc. (US) 2001-12-05 EP disclosed
WO-2001000658-A1 C-TERMINAL MODIFIED (N-SUBSTITUTED)-2-INDOLYLCARBONYLDIPEPTIDES AS INHIBITORS OF THE ICE/CED-3 FAMILY OF CYSTEINE PROTEASES IDUN PHARMACEUTICALS, INC. (US) 2001-01-04 WO disclosed