SCHEMBL7540604

SCHEMBL7540604

CCC(c1cn(Cc2ccc(OCc3csc(-c4ccccc4)n3)cc2)nc1-c1cccs1)C(CC)(C(=O)O)C(=O)O

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
RAB9A P51151 6/20 0.41
NPC1 O15118 5/20 0.41
MAPT P10636 2/20 0.41
TSHR P16473 2/20 0.41
MAPK1 P28482 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
KDM4E B2RXH2 1/20 0.39
PPARA Q07869 3/20 0.38
ALOX5 P09917 1/20 0.36
SMN1; SMN2 Q16637 4/20 0.36
TP53 P04637 2/20 0.36
NFKB1 P19838 2/20 0.36
NFKB2 Q00653 2/20 0.36
RELA Q04206 2/20 0.36
PKM P14618 1/20 0.36
HSD17B10 Q99714 1/20 0.36
KLKB1 P03952 1/20 0.36
KLK1 P06870 1/20 0.36
FFAR1 O14842 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7546664 0.88 PPARA (0.45) ALDH1A1KDM4EPPARAFFAR1PPARG
SCHEMBL7547501 0.84 PPARA (0.49) MAPTPPARAFFAR1PPARG
SCHEMBL5376653 0.83 RAB9A (0.44) ALDH1A1RAB9ANPC1MAPTTSHR
SCHEMBL7540590 0.83 RAB9A (0.43) ALDH1A1RAB9ANPC1MAPTTSHR
SCHEMBL6589744 0.83 MAPT (0.42) ALDH1A1RAB9ANPC1MAPTTSHR
SCHEMBL7543020 0.82 ALDH1A1 (0.43) ALDH1A1RAB9ANPC1MAPTTSHR
SCHEMBL5379428 0.82 RAB9A (0.46) ALDH1A1RAB9ANPC1MAPTTSHR
SCHEMBL7543023 0.81 ALDH1A1 (0.42) ALDH1A1RAB9ANPC1MAPTTSHR
SCHEMBL5372050 0.81 RAB9A (0.46) ALDH1A1RAB9ANPC1MAPTTSHR
SCHEMBL5376645 0.81 RAB9A (0.45) ALDH1A1RAB9ANPC1MAPTTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1228067-A1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGYLCEMIC AND HYPOLIPIDEMIC ACTIVITY Takeda Chemical Industries, Ltd. (JP) 2002-08-07 EP disclosed
WO-2001038325-A1 5-MEMBERED N-HETEROCYCLIC COMPOUNDS WITH HYPOGLYCEMIC AND HYPOLIPIDEMIC ACTIVITY TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-05-31 WO disclosed