SCHEMBL7540901

SCHEMBL7540901

CN1Cc2cc(NC(=O)CN(C(=O)OC(C)(C)C)c3ccccn3)ccc2CC(CC(=O)O)C1=O

nearest known ligand 0.51

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 10/20 0.51
ITGA2B P08514 9/20 0.51
ITGAV P06756 8/20 0.51
ADM2 Q7Z4H4 4/20 0.36
CALCB P10092 3/20 0.36
HDAC8 Q9BY41 2/20 0.34
CALCRL Q16602 2/20 0.34
MAP2K2 P36507 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7545780 0.79 ITGB3 (0.59) ITGB3ITGA2BITGAV
SCHEMBL7539970 0.77 ITGB3 (0.46) ITGB3ITGA2BITGAVHDAC8MAP2K2
SCHEMBL7543230 0.76 ITGB3 (0.46) ITGB3ITGA2BITGAVHDAC8
SCHEMBL7659474 0.74 ITGB3 (0.49) ITGB3ITGA2BITGAV
SCHEMBL6419667 0.73 ITGB3 (0.54) ITGB3ITGA2BITGAV
SCHEMBL6420692 0.73 ITGB3 (0.54) ITGB3ITGA2BITGAVHDAC8
SCHEMBL6418484 0.72 ITGB3 (0.70) ITGB3ITGA2BITGAV
SCHEMBL7541901 0.72 ITGB3 (0.51) ITGB3ITGA2BITGAV
SCHEMBL6418662 0.70 ITGB3 (0.51) ITGB3ITGA2BITGAV
SCHEMBL7335166 0.70 ITGB3 (0.49) ITGB3ITGA2BITGAV

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6458784-B1 PHARMACEUTICALLY ACTIVE BENZODIAZAPINE COMPOUNDS OF FORMULA (I) ARE DISCLOSED. THESE COMPOUNDS INHIBIT THE VITRONECTIN RECEPTOR AND ARE USEFUL FOR TREATMENT OF OSTEOPOROSIS. SMITHKLINE BEECHAM CORPORATION 2002-10-01 US disclosed
EP-0762882-A4 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORP (US) 2002-09-11 EP disclosed
EP-0762882-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-03-19 EP disclosed
WO-1996000574-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1996-01-11 WO disclosed