SCHEMBL7541346

SCHEMBL7541346

COC(=O)c1c(NC(=O)C(=O)OC(C)(C)C)sc2nccnc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK10 P53779 2/20 0.35
MAPK8 P45983 1/20 0.35
MAPK9 P45984 1/20 0.35
ATR Q13535 1/20 0.35
MAPT P10636 3/20 0.35
HTT P42858 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 6/20 0.33
HPGD P15428 3/20 0.33
TSHR P16473 2/20 0.33
HSD17B10 Q99714 1/20 0.33
KMT2A Q03164 2/20 0.33
CISD2 Q8N5K1 1/20 0.33
MEN1 O00255 1/20 0.33
USP2 O75604 1/20 0.33
CXCR2 P25025 1/20 0.32
PKM P14618 1/20 0.32
POLB P06746 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
TP53 P04637 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7536279 0.71 CISD2 (0.47) MAPTALDH1A1HPGDKMT2ACISD2
SCHEMBL7540301 0.68 PTPN1 (0.44)
SCHEMBL16504711 0.66 ATR (0.42) ATRMAPTHTTSMN1; SMN2ALDH1A1
SCHEMBL16504981 0.64 LCK (0.38) ATRMAPTALDH1A1HPGDTSHR
SCHEMBL18306148 0.64 ATR (0.47) MAPK10MAPK8MAPK9ATRHTT
SCHEMBL7837432 0.63 MAPT (0.38) ATRMAPTALDH1A1TSHRKMT2A
SCHEMBL16504770 0.63 LCK (0.37) ATRALDH1A1PKM
SCHEMBL4116375 0.62 KDM4E (0.50) MAPTHTTSMN1; SMN2ALDH1A1HPGD
SCHEMBL3493608 0.62 METAP1 (0.45) ATRMAPTALDH1A1HPGDKMT2A
SCHEMBL6309788 0.62 ALDH1A1 (0.39) MAPTSMN1; SMN2ALDH1A1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020019412-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPASES) NOVO NORDISK A/S (DK) 2002-02-14 US disclosed
EP-1080068-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES Novo Nordisk A/S (DK) 2001-03-07 EP disclosed
WO-1999046237-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES NOVO NORDISK A/S (DK) 1999-09-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020019412-A1 MODULATORS OF PROTEIN TYROSINE PHOSPHATASES (PTPASES) PTPRCAP, PTPRS, PTPRA MAPK10 1804/4885MAPK8 2062/4885MAPK9 2479/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.