SCHEMBL7544290

SCHEMBL7544290

N#CCNC(=O)CC(N)SCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CTSS P25774 9/20 0.46
CTSL P07711 9/20 0.46
CTSB P07858 4/20 0.46
CTSK P43235 6/20 0.45
CTSC P53634 2/20 0.43
MCL1 Q07820 1/20 0.42
ATM Q13315 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5526400 0.78 CTSS (0.44) CTSSCTSLCTSBCTSK
SCHEMBL6467489 0.76 CYP2C19 (0.46)
SCHEMBL7544294 0.75 CTSC (0.51) CTSSCTSLCTSBCTSKCTSC
Hydrochloric Acid SCHEMBL6467921 0.75 IDO1 (0.45)
SCHEMBL6742393 0.74 CTSS (0.49) CTSSCTSLCTSBCTSKATM
SCHEMBL3622046 0.73 CTSS (0.41) CTSSCTSLCTSBCTSK
SCHEMBL10612693 0.73 CTSS (0.66) CTSSCTSLCTSBCTSKMCL1
SCHEMBL5524114 0.71 CTSL (0.56) CTSSCTSLCTSBCTSK
SCHEMBL16626138 0.71 CTSS (0.67) CTSSCTSLCTSBCTSKCTSC
SCHEMBL5456972 0.71 CTSS (0.67) CTSSCTSLCTSBCTSKCTSC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1212302-A1 COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2002-06-12 EP disclosed
WO-2001019796-A1 COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS AS CATHEPSIN S INHIBITORS AXYS PHARMACEUTICALS, INC. (US) 2001-03-22 WO disclosed