SCHEMBL7544343

SCHEMBL7544343

COc1ccc(CN2C(=O)C(F)(F)C2C(=O)OCC(C)C)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.40
PKM P14618 1/20 0.40
KDM4E B2RXH2 3/20 0.39
KMT2A Q03164 3/20 0.39
LMNA P02545 2/20 0.39
CMA1 P23946 1/20 0.39
ALDH1A1 P00352 3/20 0.38
CYP3A4 P08684 1/20 0.38
GSK3A P49840 1/20 0.37
GSK3B P49841 1/20 0.37
HKDC1 Q2TB90 1/20 0.37
MEN1 O00255 2/20 0.37
TSHR P16473 1/20 0.36
ANPEP P15144 1/20 0.36
HPGD P15428 1/20 0.36
HDAC3 O15379 1/20 0.36
HDAC4 P56524 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC7 Q8WUI4 1/20 0.36
HDAC2 Q92769 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7544337 1.00 POLB (0.40) POLBPKMKDM4EKMT2ALMNA
SCHEMBL10323975 0.71 MEN1 (0.54) POLBKMT2ACMA1ALDH1A1GSK3B
SCHEMBL22287862 0.70 MMP1 (0.42) KDM4EKMT2ACMA1ALDH1A1CYP3A4
SCHEMBL22287726 0.68 TP53 (0.51) KDM4EKMT2ALMNAALDH1A1HKDC1
SCHEMBL31404224 0.66 CYP3A4 (0.40) POLBKDM4ELMNACMA1CYP3A4
SCHEMBL21847080 0.66 KDM4E (0.51) KDM4EKMT2ALMNACMA1ALDH1A1
SCHEMBL25316050 0.65 ALDH1A1 (0.43) POLBPKMKDM4EKMT2AALDH1A1
SCHEMBL30714028 0.64 GAA (0.49) KDM4EKMT2ACMA1ALDH1A1CYP3A4
SCHEMBL430661 0.64 CMA1 (0.66) KDM4EKMT2ACMA1ALDH1A1GSK3A
SCHEMBL25894467 0.64 ALDH1A1 (0.42) KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2002045853-A1 LEWIS ACID CATALYSIS USING CHIRAL METAL COMPLEXES DOYLE MICHAEL P (US) 2002-06-13 WO disclosed