SCHEMBL7544931

SCHEMBL7544931

OC[C@@H](O)c1cncc(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCAR2 Q8TDS4 1/20 0.39
PYGL P06737 3/20 0.36
GRIN1 Q05586 1/20 0.34
GRIN2B Q13224 1/20 0.34
CYP3A4 P08684 1/20 0.33
TSHR P16473 1/20 0.33
P2RX7 Q99572 1/20 0.33
TRPV3 Q8NET8 1/20 0.33
CHRNB2 P17787 2/20 0.33
CHRNA4 P43681 2/20 0.33
MKNK1 Q9BUB5 1/20 0.33
MKNK2 Q9HBH9 1/20 0.33
ICAM1 P05362 1/20 0.32
SELE P16581 1/20 0.32
VCAM1 P19320 1/20 0.32
ADORA3 P0DMS8 2/20 0.32
ADORA1 P30542 2/20 0.32
ADORA2A P29274 1/20 0.32
ADORA2B P29275 1/20 0.32
SCN9A Q15858 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30527645 0.86 BLM (0.41) HCAR2CYP3A4TSHRMKNK1MKNK2
SCHEMBL25261700 0.86 BLM (0.41) HCAR2CYP3A4TSHRMKNK1MKNK2
SCHEMBL20832851 0.86 HCAR2 (0.38) HCAR2GRIN1GRIN2BP2RX7CHRNB2
SCHEMBL20832745 0.86 HCAR2 (0.38) HCAR2GRIN1GRIN2BP2RX7CHRNB2
SCHEMBL20832746 0.84 LMNA (0.41) HCAR2GRIN1GRIN2BP2RX7TRPV3
SCHEMBL19895723 0.80 HCAR2 (0.34) HCAR2GRIN1GRIN2BP2RX7CHRNB2
SCHEMBL20292644 0.77 GAA (0.35) HCAR2GRIN1GRIN2BCYP3A4ADORA3
SCHEMBL25308368 0.77 ALDH1A1 (0.46) HCAR2TSHRP2RX7MKNK1MKNK2
SCHEMBL31250294 0.77 ALDH1A1 (0.46) HCAR2TSHRP2RX7MKNK1MKNK2
SCHEMBL16491297 0.77 CYP11B2 (0.41) HCAR2TRPV3CHRNB2CHRNA4MKNK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1175416-A1 HETEROARYL DIAZACYCLOALKANES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 2002-01-30 EP disclosed
WO-2000064885-A1 HETEROARYL DIAZACYCLOALKANES, THEIR PREPARATION AND USE NEUROSEARCH A/S (DK) 2000-11-02 WO disclosed