SCHEMBL754554

SCHEMBL754554

O=CCCCCC1CCSS1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 2/20 0.58
KMT2A Q03164 2/20 0.58
TARDBP Q13148 2/20 0.58
CYP2C9 P11712 1/20 0.58
MEN1 O00255 1/20 0.58
NR1I2 O75469 1/20 0.58
ALDH1A1 P00352 1/20 0.58
LMNA P02545 1/20 0.58
POLB P06746 1/20 0.58
THRB P10828 1/20 0.58
TSHR P16473 1/20 0.58
ACHE P22303 1/20 0.58
APEX1 P27695 1/20 0.58
RECQL P46063 1/20 0.58
BLM P54132 1/20 0.58
PMP22 Q01453 1/20 0.58
TDP1 Q9NUW8 1/20 0.58
SAE1 Q9UBE0 1/20 0.58
UBA2 Q9UBT2 1/20 0.58
L3MBTL1 Q9Y468 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8521624 1.00 HSD17B10 (0.58) HSD17B10KMT2ATARDBPCYP2C9MEN1
SCHEMBL29249729 0.98 HSD17B10 (0.56) HSD17B10KMT2ATARDBPCYP2C9MEN1
SCHEMBL29249658 0.98 HSD17B10 (0.56) HSD17B10KMT2ATARDBPCYP2C9MEN1
SCHEMBL16053552 0.96 HSD17B10 (0.54) HSD17B10KMT2ATARDBPCYP2C9MEN1
SCHEMBL29263924 0.85 HSD17B10 (0.67) HSD17B10KMT2ATARDBPCYP2C9MEN1
SCHEMBL19160682 0.80 HSD17B10 (0.53) HSD17B10KMT2ATARDBPCYP2C9MEN1
SCHEMBL8516674 0.79 CA12 (0.62) HSD17B10KMT2ATARDBPCYP2C9MEN1
SCHEMBL16144543 0.78 HSD17B10 (0.51) HSD17B10KMT2ATARDBPCYP2C9MEN1
SCHEMBL17612125 0.78 HSD17B10 (0.51) HSD17B10KMT2ATARDBPCYP2C9MEN1
SCHEMBL15182687 0.77 HSD17B10 (0.54) HSD17B10KMT2ATARDBPCYP2C9MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2621537-B1 PENTAPEPTIDE DERIVATIVES FOR PROMOTING HAIR GROWTH ELFETIN COSMETICS AG (CH) 2015-02-25 EP claimed
US-20130209551-A1 PENTAPEPTIDE DERIVATIVES FOR PROMOTING HAIR GROWTH ELFETIN COSMETICS AG (CH) 2013-08-15 US claimed
US-20090285888-A1 DERIVATIVES OF DIHYDROXYPHENYLALANINE ELLNEUROXX LTD. (DE) 2009-11-19 US claimed
CN-101208326-A Derivate von dihydroxyphenylalanin ELLNEUROXX LTD (DE) 2008-06-25 CN claimed
EP-4282411-A1 LIPOYL-GLU-ALA FOR THE TREATMENT OF NEURODEGENERATIVE DAMAGE CAUSED BY TRAUMATIC BRAIN INJURY Ischemix LLC (US) 2023-11-29 EP disclosed
EP-2804862-B1 METHODS OF MAKING AND USING NANOSTRUCTURES UNIV MINNESOTA (US) 2019-07-17 EP disclosed
US-10239906-B2 Apparatus and method for obtaining glycoglycerolipids and glycosphingolipids from lipid phases NANOSCIENCE FOR LIFE GMBH & COKG (DE) 2019-03-26 US disclosed
EP-3152219-B1 METHOD FOR OBTAINING GLYCOGLYCEROLIPIDS AND GLYCOSPHINGOLIPIDS FROM LIPOID PHASES NANOSCIENCE FOR LIFE GMBH & CO KG (DE) 2019-01-09 EP disclosed
WO-2018053706-A1 COMPOSITION COMPRISING PAEONIFLORIN OR ALBIFLORIN ANALOGUE, METHOD OF PREPARATION THEREOF L'OREAL (FR) 2018-03-29 WO disclosed
EP-2640423-B1 LIPOYL COMPOUNDS AND THEIR USE FOR TREATING ISCHEMIC INJURY ISCHEMIX LLC (US) 2017-07-26 EP disclosed
US-20170121360-A1 APPARATUS AND METHOD FOR OBTAINING GLYCOGLYCEROLIPIDS AND GLYCOSPHINGOLIPIDS FROM LIPID PHASES GEA WESTFALIA SEPARATOR GROUP GMBH (DE) 2017-05-04 US disclosed
US-9540417-B2 Compositions and methods for treating ischemia and ischemia-reperfusion injury ISCHEMIX LLC (US) 2017-01-10 US disclosed
US-20090285888-A1 DERIVATIVES OF DIHYDROXYPHENYLALANINE ELLNEUROXX LTD. (DE) 2009-11-19 US disclosed
US-20090117346-A1 PHOTOSENSITIVE MATERIAL FOR FORMING CONDUCTIVE FILM, CONDUCTIVE FILM, LIGHT TRANSMITTING ELECTROMAGNETIC WAVE SHIELDING FILM AND METHOD FOR MANUFACTURING THE SAME FUJIFILM CORPORATION (JP) 2009-05-07 US disclosed
US-20090098480-A1 PHOTOSENSITIVE MATERIAL FOR FORMING CONDUCTIVE FILM, CONDUCTIVE FILM, LIGHT TRANSMITTING ELECTROMAGNETIC WAVE SHIELDING FILM AND METHOD FOR MANUFACTURING THE SAME FUJIFILM CORPORATION (JP) 2009-04-16 US disclosed
US-20090098481-A1 PHOTOSENSITIVE MATERIAL FOR FORMING CONDUCTIVE FILM, CONDUCTIVE FILM, LIGHT TRANSMITTING ELECTROMAGNETIC WAVE SHIELDING FILM AND METHOD FOR MANUFACTURING THE SAME FUJIFILM CORPORATION (JP) 2009-04-16 US disclosed
US-20090029125-A1 PHOTOSENSITIVE MATERIAL FOR FORMING CONDUCTIVE FILM, CONDUCTIVE FILM, LIGHT TRANSMITTING ELECTROMAGNETIC WAVE SHIELDING FILM AND METHOD FOR MANUFACTURING THE SAME FUJIFILM CORPORATION (JP) 2009-01-29 US disclosed
CN-101208326-A Derivate von dihydroxyphenylalanin ELLNEUROXX LTD (DE) 2008-06-25 CN disclosed
US-7320867-B2 Linker compound, ligand, and producing method thereof JAPAN SCIENCE AND TECHNOLOGY AGENCY (JP) 2008-01-22 US disclosed
WO-2006021413-A1 ALPHA-KETO CARBONYL CALPAIN INHIBITORS SANTHERA PHARMACEUTICALS (SCHWEIZ) AG (CH) 2006-03-02 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090285888-A1 DERIVATIVES OF DIHYDROXYPHENYLALANINE HTT, NLN, SNCA HSD17B10 1148/4885KMT2A 717/4885TARDBP 27/4885
US-20130209551-A1 PENTAPEPTIDE DERIVATIVES FOR PROMOTING HAIR GROWTH NGLY1, CCNA1, TOE1 HSD17B10 846/4885KMT2A 2749/4885TARDBP 4352/4885
US-20170121360-A1 APPARATUS AND METHOD FOR OBTAINING GLYCOGLYCEROLIPIDS AND GLYCOSPHINGOLIPIDS FROM LIPID PHASES AGL, LIPA, MGLL HSD17B10 348/4885KMT2A 2643/4885TARDBP 4871/4885
US-10239906-B2 Apparatus and method for obtaining glycoglycerolipids and glycosphingolipids from lipid phases AGL, LIPA, MGLL HSD17B10 348/4885KMT2A 2643/4885TARDBP 4871/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.