SCHEMBL7545918

SCHEMBL7545918

CC(O)CC=Cc1cccc(N(C)C)c1

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
TSHR P16473 1/20 0.41
NPC1 O15118 1/20 0.40
MAPT P10636 1/20 0.40
MAPK1 P28482 1/20 0.40
RAB9A P51151 1/20 0.40
HTR2A P28223 3/20 0.40
APP P05067 3/20 0.40
NR1H4 Q96RI1 2/20 0.38
HDAC4 P56524 1/20 0.38
MEF2D Q14814 1/20 0.38
GSK3B P49841 1/20 0.37
RELA Q04206 1/20 0.36
EPOR P19235 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7545910 1.00 ALDH1A1 (0.41) ALDH1A1TSHRNPC1MAPTMAPK1
SCHEMBL7546223 0.82 CHRNB2 (0.54) ALDH1A1TSHRNPC1MAPTMAPK1
SCHEMBL7546225 0.82 CHRNB2 (0.54) ALDH1A1TSHRNPC1MAPTMAPK1
SCHEMBL13703007 0.78 HTR2A (0.42) ALDH1A1TSHRMAPTHTR2AHDAC4
SCHEMBL6258001 0.78 CYP19A1 (0.50) NPC1MAPTHTR2A
SCHEMBL6258006 0.78 CYP19A1 (0.50) NPC1MAPTHTR2A
SCHEMBL13703006 0.78 HTR2A (0.42) ALDH1A1TSHRMAPTHTR2AHDAC4
SCHEMBL13703292 0.76 HDAC4 (0.41) ALDH1A1HTR2AHDAC4MEF2DEPOR
SCHEMBL13703318 0.76 HDAC4 (0.41) ALDH1A1HTR2AHDAC4MEF2DEPOR
SCHEMBL5475692 0.76 HTR2A (0.66) TSHRHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1214288-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE Targacept Inc. (US) 2002-06-19 EP disclosed
US-6337351-B1 AROMATIC OLEFIN AMINES TARGACEPT, INC. 2002-01-08 US disclosed
WO-2001017943-A1 PHARMACEUTICAL COMPOSITIONS AND METHODS FOR USE TARGACEPT, INC. (US) 2001-03-15 WO disclosed