SCHEMBL7546209

SCHEMBL7546209

CCn1nc(Cc2ccccc2)cc1C1CCN(OC(=O)C(F)(F)F)CC1

nearest known ligand 0.51

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 20/20 0.51
KCNH2 Q12809 4/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27643633 0.83 CCR5 (0.49) CCR5KCNH2
SCHEMBL5451783 0.82 CCR5 (0.54) CCR5KCNH2
Trifluoroacetic Acid SCHEMBL5764463 0.81 CCR5 (0.49) CCR5KCNH2
Trifluoroacetic Acid SCHEMBL7546206 0.81 CCR5 (0.49) CCR5KCNH2
SCHEMBL27643626 0.79 CCR5 (0.49) CCR5KCNH2
SCHEMBL7502186 0.78 CCR5 (0.47) CCR5
SCHEMBL7547218 0.77 LCK (0.42)
SCHEMBL5456417 0.74 CCR5 (0.48) CCR5KCNH2
SCHEMBL5456416 0.74 CCR5 (0.51) CCR5KCNH2
Hydrochloric Acid SCHEMBL5764233 0.73 GABRA1 (0.48) CCR5KCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1171122-A4 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO INC (US) 2002-05-29 EP disclosed
EP-1171122-A1 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY Merck & Co., Inc. (US) 2002-01-16 EP disclosed
US-6248755-B1 ANTIINFLAMMATORY AGENTS; ANTIALLERGENS; AUTOIMMUNE DISEASES MERCK & CO., INC. 2001-06-19 US disclosed
WO-2000059502-A1 PYRROLIDINE MODULATORS OF CHEMOKINE RECEPTOR ACTIVITY MERCK & CO., INC. (US) 2000-10-12 WO disclosed