SCHEMBL7546623

SCHEMBL7546623

COc1cc(Br)c(OC)c2c1CC(NC=O)CC2

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 4/20 0.45
CYP1A2 P05177 1/20 0.37
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
PRKDC P78527 1/20 0.35
CA1 P00915 2/20 0.34
CA2 P00918 2/20 0.34
CA4 P22748 1/20 0.34
CA6 P23280 1/20 0.34
DRD2 P14416 1/20 0.34
DRD4 P21917 1/20 0.34
DRD3 P35462 1/20 0.34
MTNR1A P48039 4/20 0.34
MTNR1B P49286 4/20 0.34
MEN1 O00255 1/20 0.33
TNF P01375 1/20 0.33
KMT2A Q03164 1/20 0.33
NOD2 Q9HC29 1/20 0.33
NOD1 Q9Y239 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7542176 0.95 HTR2A (0.45) HTR2ACYP1A2MAPTHPGDPRKDC
SCHEMBL7548050 0.84 HTR2A (0.49) HTR2ACYP1A2CA1CA2CA4
Hydrochloric Acid SCHEMBL7540742 0.83 HTR2A (0.48) HTR2ACYP1A2MAPTCA1CA2
SCHEMBL7544348 0.82 CYP1A2 (0.56) CYP1A2MAPTCA1CA2DRD2
Hydrochloric Acid SCHEMBL7547168 0.77 HTR2A (0.48) HTR2ACYP1A2MAPTCA1CA2
SCHEMBL7544871 0.75 ADRA1A (0.59) HTR2ACYP1A2DRD2DRD3ADRA1A
SCHEMBL7541153 0.72 ADRA1A (0.41) CYP1A2MAPTCA1CA2DRD2
SCHEMBL7543110 0.72 ADRA1A (0.44) CYP1A2MAPTDRD2DRD4DRD3
SCHEMBL11299373 0.71 HTR2A (0.50) HTR2ACYP1A2CA1CA2CA4
SCHEMBL7540836 0.70 MTNR1A (0.65) CYP1A2MAPTDRD2DRD4DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0883599-B1 AMINOTETRALIN DERIVATIVES AND COMPOSITIONS AND METHOD OF USE THEREOF ASTRAZENECA AB (SE) 2002-06-05 EP disclosed
EP-0883599-A1 AMINOTETRALIN DERIVATIVES AND COMPOSITIONS AND METHOD OF USE THEREOF ZENECA LIMITED (GB) 1998-12-16 EP disclosed
US-5807897-A MUSCULAR DISORDERS ZENECA LIMITED (GB) 1998-09-15 US disclosed
WO-1997031887-A1 AMINOTETRALIN DERIVATIVES AND COMPOSITIONS AND METHOD OF USE THEREOF ZENECA LIMITED (GB) 1997-09-04 WO disclosed