SCHEMBL7547648

SCHEMBL7547648

CC(CN(C)C)n1cc(-c2cncc(-c3ccsc3)c2)c2ccc(Cl)cc21

nearest known ligand 0.58

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.58
FLT1 P17948 4/20 0.58
FLT4 P35916 4/20 0.58
CYP2A6 P11509 4/20 0.40
TDP2 O95551 1/20 0.36
NFATC1 O95644 1/20 0.34
GSK3B P49841 1/20 0.34
DYRK1A Q13627 1/20 0.34
CHEK2 O96017 1/20 0.33
PIK3CD O00329 1/20 0.33
CYP11B1 P15538 1/20 0.31
CYP11B2 P19099 1/20 0.31
GAK O14976 1/20 0.30
HTR1D P28221 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7550794 0.92 KDR (0.56) KDRFLT1FLT4CYP2A6TDP2
SCHEMBL7976277 0.88 KDR (0.43) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7551876 0.87 KDR (0.72) KDRFLT1FLT4CYP2A6NFATC1
SCHEMBL7557902 0.86 KDR (0.46) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7988607 0.85 KDR (0.43) KDRFLT1FLT4NFATC1GSK3B
SCHEMBL7988018 0.85 KDR (0.78) KDRFLT1FLT4CYP2A6TDP2
SCHEMBL7990418 0.83 KDR (0.39) KDRFLT1FLT4CYP11B1CYP11B2
SCHEMBL7553622 0.82 KDR (0.55) KDRFLT1FLT4CYP2A6TDP2
SCHEMBL7991178 0.81 KDR (0.54) KDRFLT1FLT4CYP2A6
SCHEMBL7976429 0.79 KDR (0.78) KDRFLT1FLT4CYP2A6TDP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147107-A4 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO INC (US) 2002-05-22 EP claimed
EP-1147107-A1 NOVEL ANGIOGENESIS INHIBITORS Merck & Co., Inc. (US) 2001-10-24 EP claimed
US-6281389-B1 MIXING WITH SOLVENT; DISTILLATION NIPPON SHOKUBAI CO., LTD. (JP) 2001-08-28 US claimed
WO-2000043393-A1 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO., INC. (US) 2000-07-27 WO claimed
EP-1147107-A4 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO INC (US) 2002-05-22 EP disclosed
EP-1147107-A1 NOVEL ANGIOGENESIS INHIBITORS Merck & Co., Inc. (US) 2001-10-24 EP disclosed
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed
WO-2000043393-A1 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO., INC. (US) 2000-07-27 WO disclosed