SCHEMBL7990418

SCHEMBL7990418

COc1ccc(-c2cncc(-c3cn(C(C)CN(C)C)c4cc(Cl)ccc34)c2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.39
FLT1 P17948 1/20 0.39
FLT4 P35916 1/20 0.39
ALPL P05186 1/20 0.39
BMP4 P12644 1/20 0.38
MAP4K4 O95819 1/20 0.35
CYP19A1 P11511 3/20 0.35
PDE4B Q07343 1/20 0.35
PDE4D Q08499 1/20 0.35
NLRP3 Q96P20 1/20 0.35
CYP11B1 P15538 3/20 0.34
CYP11B2 P19099 3/20 0.34
CYP17A1 P05093 1/20 0.34
ADORA3 P0DMS8 1/20 0.34
ADORA1 P30542 1/20 0.34
MAT2A P31153 1/20 0.33
AURKA O14965 1/20 0.33
AURKB Q96GD4 1/20 0.33
CHEK1 O14757 1/20 0.33
CYP3A4 P08684 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7976277 0.92 KDR (0.43) KDRFLT1FLT4ALPLMAP4K4
SCHEMBL7987876 0.89 PDE4B (0.45) KDRFLT1FLT4ALPLPDE4B
SCHEMBL7557902 0.88 KDR (0.46) KDRFLT1FLT4CYP11B1CYP11B2
SCHEMBL7550587 0.87 KDR (0.49) KDRFLT1FLT4BMP4MAP4K4
SCHEMBL7549809 0.86 HTR6 (0.43) KDRFLT1FLT4ALPLMAP4K4
SCHEMBL7988607 0.85 KDR (0.43) KDRFLT1FLT4CYP11B1CYP11B2
SCHEMBL7552885 0.83 KDR (0.51) KDRFLT1FLT4MAP4K4PDE4B
SCHEMBL7547648 0.83 KDR (0.58) KDRFLT1FLT4CYP11B1CYP11B2
SCHEMBL7976435 0.82 PRKCA (0.42) KDRFLT1FLT4ALPLPDE4B
SCHEMBL7990227 0.82 PDE4B (0.45) KDRFLT1FLT4PDE4BPDE4D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed