SCHEMBL7988018

SCHEMBL7988018

CC(CN(C)C)Cn1cc(-c2cncc(-c3ccsc3)c2)c2ccc(Cl)cc21

nearest known ligand 0.78

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KDR P35968 8/20 0.78
FLT1 P17948 4/20 0.78
FLT4 P35916 4/20 0.78
CYP2A6 P11509 4/20 0.39
KCNH2 Q12809 1/20 0.38
DYRK1A Q13627 1/20 0.38
TDP2 O95551 1/20 0.35
PRKACA P17612 1/20 0.34
PRKACG P22612 1/20 0.34
PRKACB P22694 1/20 0.34
PIK3CD O00329 1/20 0.32
CHEK2 O96017 1/20 0.32
MAPK1 P28482 1/20 0.32
HTR1D P28221 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7976429 0.93 KDR (0.78) KDRFLT1FLT4CYP2A6KCNH2
SCHEMBL7548685 0.88 KDR (0.60) KDRFLT1FLT4KCNH2DYRK1A
SCHEMBL7547755 0.88 KDR (1.00) KDRFLT1FLT4CYP2A6KCNH2
SCHEMBL7990966 0.87 KDR (0.63) KDRFLT1FLT4KCNH2DYRK1A
SCHEMBL7508525 0.86 KDR (0.59) KDRFLT1FLT4KCNH2DYRK1A
SCHEMBL7547648 0.85 KDR (0.58) KDRFLT1FLT4CYP2A6DYRK1A
SCHEMBL7551687 0.83 KDR (0.77) KDRFLT1FLT4CYP2A6TDP2
SCHEMBL7987137 0.83 KDR (0.74) KDRFLT1FLT4CYP2A6KCNH2
SCHEMBL7550053 0.82 KDR (0.75) KDRFLT1FLT4CYP2A6KCNH2
SCHEMBL7505482 0.81 KDR (0.54) KDRFLT1FLT4KCNH2DYRK1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed