SCHEMBL7550287

SCHEMBL7550287

CN(C)CCn1cc(-c2cncc(-c3ccsc3)c2)c2ccccc21

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDR P35968 9/20 1.00
FLT1 P17948 4/20 0.72
FLT4 P35916 4/20 0.72
HTR1D P28221 1/20 0.47
CYP2A6 P11509 2/20 0.45
GSK3B P49841 1/20 0.44
HTR6 P50406 4/20 0.42
PRKCB P05771 2/20 0.41
PRKCA P17252 2/20 0.41
PRKCH P24723 1/20 0.39
PRKCE Q02156 1/20 0.39
PRKCQ Q04759 1/20 0.39
PRKCD Q05655 1/20 0.39
FLT3 P36888 1/20 0.39
CNR2 P34972 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7553991 0.94 KDR (1.00) KDRFLT1FLT4CYP2A6GSK3B
SCHEMBL7549872 0.90 KDR (0.81) KDRFLT1FLT4HTR1DCYP2A6
SCHEMBL7554970 0.90 KDR (0.81) KDRFLT1FLT4HTR1DCYP2A6
SCHEMBL7551626 0.88 KDR (0.79) KDRFLT1FLT4HTR1DCYP2A6
SCHEMBL7550368 0.85 KDR (0.73) KDRFLT1FLT4CYP2A6HTR6
SCHEMBL7547755 0.84 KDR (1.00) KDRFLT1FLT4HTR1DCYP2A6
SCHEMBL7555190 0.82 KDR (1.00) KDRFLT1FLT4CYP2A6GSK3B
SCHEMBL7976107 0.82 KDR (0.68) KDRFLT1FLT4CYP2A6GSK3B
SCHEMBL7556531 0.81 KDR (1.00) KDRFLT1FLT4CYP2A6GSK3B
SCHEMBL7549908 0.81 KDR (1.00) KDRFLT1FLT4CYP2A6GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147107-A4 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO INC (US) 2002-05-22 EP claimed
EP-1147107-A1 NOVEL ANGIOGENESIS INHIBITORS Merck & Co., Inc. (US) 2001-10-24 EP claimed
WO-2000043393-A1 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO., INC. (US) 2000-07-27 WO claimed
EP-1147107-A4 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO INC (US) 2002-05-22 EP disclosed
EP-1147107-A1 NOVEL ANGIOGENESIS INHIBITORS Merck & Co., Inc. (US) 2001-10-24 EP disclosed
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed
WO-2000043393-A1 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO., INC. (US) 2000-07-27 WO disclosed