SCHEMBL7552049

SCHEMBL7552049

c1ccc(CNCC2CCCN2Cc2ccccc2)cc1

nearest known ligand 0.56

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
CXCR4 P61073 2/20 0.56
OPRL1 P41146 1/20 0.49
CCR2 P41597 3/20 0.48
SPHK2 Q9NRA0 2/20 0.47
SPHK1 Q9NYA1 2/20 0.47
KDM4E B2RXH2 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6541445 0.95 CXCR4 (0.55) CXCR4OPRL1CCR2
SCHEMBL6541449 0.95 CXCR4 (0.55) CXCR4OPRL1CCR2
SCHEMBL11419710 0.87 KDM4E (0.59) CXCR4KDM4E
SCHEMBL11462791 0.86 CCR2 (0.49) CCR2SPHK2SPHK1
SCHEMBL11459718 0.82 CCR2 (0.49) CCR2SPHK2SPHK1
SCHEMBL7454601 0.82 OPRD1 (0.52) CCR2
SCHEMBL16293069 0.81 CXCR4 (0.47) CXCR4OPRL1CCR2SPHK2SPHK1
SCHEMBL14454201 0.81 CCR2 (0.48) CCR2SPHK2SPHK1
SCHEMBL13220244 0.80 CXCR4 (0.50) CXCR4
SCHEMBL19946919 0.79 CCR2 (0.61) CCR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1137412-A4 SUBSTITUTED NITROGEN HETEROCYCLIC COMPOUNDS AND THERAPEUTIC USES THEREOF AMERICAN BIOGENETIC SCIENCES (US) 2002-04-03 EP disclosed
EP-1137412-A2 SUBSTITUTED NITROGEN HETEROCYCLIC COMPOUNDS AND THERAPEUTIC USES THEREOF AMERICAN BIOGENETIC SCIENCES, INC. (US) 2001-10-04 EP disclosed
WO-2000033788-A2 SUBSTITUTED NITROGEN HETEROCYCLIC COMPOUNDS AND THERAPEUTIC USES THEREOF AMERICAN BIOGENETIC SCIENCES INC. (US) 2000-06-15 WO disclosed