SCHEMBL7555128

SCHEMBL7555128

C=CCC1(c2ccc(Cl)c(Cl)c2)CCC(=O)N(C2CCCCC2)C1

nearest known ligand 0.59

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
TACR1 P25103 11/20 0.59
TACR2 P21452 8/20 0.45
SLC6A4 P31645 2/20 0.40
SLC6A3 Q01959 2/20 0.40
SLC6A2 P23975 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7555122 1.00 TACR1 (0.59) TACR1TACR2SLC6A4SLC6A3SLC6A2
SCHEMBL6984664 0.80 TACR1 (0.61) TACR1TACR2
SCHEMBL7566317 0.79 TACR2 (0.60) TACR1TACR2SLC6A4SLC6A3SLC6A2
SCHEMBL7566323 0.79 TACR2 (0.60) TACR1TACR2SLC6A4SLC6A3SLC6A2
SCHEMBL7134657 0.75 TACR1 (0.44) TACR1TACR2SLC6A4SLC6A3SLC6A2
SCHEMBL7134653 0.75 TACR1 (0.44) TACR1TACR2SLC6A4SLC6A3SLC6A2
SCHEMBL6968576 0.71 TACR1 (0.45) TACR1TACR2
SCHEMBL22917998 0.69 SLC6A4 (0.46) SLC6A4SLC6A3SLC6A2
SCHEMBL6950674 0.69 BACE1 (0.45) SLC6A4SLC6A3SLC6A2
SCHEMBL20457210 0.67 SLC6A4 (0.46) SLC6A4SLC6A3SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0888337-B1 PIPERIDONE TACHYKININ ANTAGONISTS PFIZER RES & DEV (IE) 2002-06-05 EP disclosed
US-6262075-B1 Piperidone tachykinin antagonists PFIZER INC 2001-07-17 US disclosed