SCHEMBL7555367

SCHEMBL7555367

COc1cccc(-c2cncc(-c3cn(CCCN4CCCCC4)c4c(OC)cccc34)c2)c1

nearest known ligand 0.51

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.51
FLT1 P17948 2/20 0.51
FLT4 P35916 2/20 0.51
CNR2 P34972 2/20 0.47
HRH3 Q9Y5N1 4/20 0.42
KDM4E B2RXH2 1/20 0.42
ALDH1A1 P00352 1/20 0.42
KMT2A Q03164 1/20 0.42
ACP1 P24666 1/20 0.41
KCNH2 Q12809 2/20 0.40
GSK3B P49841 3/20 0.40
QPCT Q16769 3/20 0.40
BACE1 P56817 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7988115 0.95 KDR (0.49) KDRFLT1FLT4CNR2HRH3
SCHEMBL7556041 0.93 KDR (0.53) KDRFLT1FLT4CNR2ALDH1A1
SCHEMBL7549404 0.92 KDR (0.51) KDRFLT1FLT4CNR2HRH3
SCHEMBL7550389 0.92 KDR (0.55) KDRFLT1FLT4CNR2HRH3
SCHEMBL7553648 0.90 KDR (0.50) KDRFLT1FLT4CNR2HRH3
SCHEMBL7554716 0.88 KDR (0.51) KDRFLT1FLT4CNR2HRH3
SCHEMBL7549925 0.87 KDR (0.67) KDRFLT1FLT4HRH3ACP1
SCHEMBL7976879 0.86 KDR (0.50) KDRFLT1FLT4CNR2ALDH1A1
SCHEMBL7549676 0.86 KDR (0.50) KDRFLT1FLT4CNR2HRH3
SCHEMBL7551199 0.86 KDR (0.54) KDRFLT1FLT4CNR2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147107-A4 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO INC (US) 2002-05-22 EP disclosed
EP-1147107-A1 NOVEL ANGIOGENESIS INHIBITORS Merck & Co., Inc. (US) 2001-10-24 EP disclosed
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed
WO-2000043393-A1 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO., INC. (US) 2000-07-27 WO disclosed