SCHEMBL7988115

SCHEMBL7988115

COc1cccc(-c2cncc(-c3cn(CCN4CCCCC4)c4c(OC)cccc34)c2)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 4/20 0.49
CNR2 P34972 1/20 0.44
FLT1 P17948 2/20 0.44
FLT4 P35916 2/20 0.44
BACE1 P56817 1/20 0.40
FLT3 P36888 1/20 0.40
BRD4 O60885 1/20 0.40
HRH3 Q9Y5N1 3/20 0.39
CYP11B1 P15538 1/20 0.39
CYP11B2 P19099 1/20 0.39
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39
LMNA P02545 2/20 0.39
ACP1 P24666 1/20 0.39
LTA4H P09960 1/20 0.39
TP53 P04637 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7555367 0.95 KDR (0.51) KDRCNR2FLT1FLT4BACE1
SCHEMBL7976879 0.92 KDR (0.50) KDRCNR2FLT1FLT4ALDH1A1
SCHEMBL7549676 0.92 KDR (0.50) KDRCNR2FLT1FLT4FLT3
SCHEMBL7551199 0.92 KDR (0.54) KDRCNR2FLT1FLT4BACE1
SCHEMBL7550092 0.90 KDR (0.49) KDRCNR2FLT1FLT4FLT3
SCHEMBL7556041 0.87 KDR (0.53) KDRCNR2FLT1FLT4BRD4
SCHEMBL7550119 0.87 CNR2 (0.40) KDRCNR2FLT1FLT4BRD4
SCHEMBL7554271 0.87 KDR (0.49) KDRCNR2FLT1FLT4FLT3
SCHEMBL7554226 0.87 KDR (0.66) KDRFLT1FLT4BACE1FLT3
SCHEMBL7549404 0.86 KDR (0.51) KDRCNR2FLT1FLT4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6265403-B1 TYROSINE INHIBITORS MERCK & CO., INC. 2001-07-24 US disclosed