SCHEMBL7555418

SCHEMBL7555418

COC(=O)c1cccc2c1c(-c1cncc(-c3ccc(Cl)cc3)c1)cn2CCCN1CCCCC1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KDR P35968 3/20 0.47
FLT1 P17948 2/20 0.47
FLT4 P35916 2/20 0.47
SMYD2 Q9NRG4 3/20 0.44
GSK3B P49841 4/20 0.39
QPCT Q16769 4/20 0.39
NR3C1 P04150 1/20 0.39
HRH3 Q9Y5N1 4/20 0.38
MEN1 O00255 1/20 0.38
GAA P10253 1/20 0.38
KMT2A Q03164 1/20 0.38
AVPR1B P47901 1/20 0.38
CHRNA7 P36544 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7987156 0.95 KDR (0.46) KDRFLT1FLT4SMYD2MEN1
SCHEMBL7551283 0.93 KDR (0.49) KDRFLT1FLT4SMYD2GSK3B
SCHEMBL7987672 0.93 KDR (0.47) KDRFLT1FLT4SMYD2HRH3
SCHEMBL7549576 0.93 KDR (0.51) KDRFLT1FLT4SMYD2GSK3B
SCHEMBL7551275 0.92 KDR (0.47) KDRFLT1FLT4SMYD2GSK3B
SCHEMBL7549814 0.88 FLT1 (0.47) KDRFLT1FLT4SMYD2HRH3
SCHEMBL7993627 0.88 KDR (0.45) KDRFLT1FLT4SMYD2HRH3
SCHEMBL7991040 0.88 FLT1 (0.47) KDRFLT1FLT4NR3C1
SCHEMBL7554912 0.87 KDR (0.50) KDRFLT1FLT4SMYD2HRH3
SCHEMBL7549476 0.87 KDR (0.65) KDRFLT1FLT4SMYD2GSK3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1147107-A4 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO INC (US) 2002-05-22 EP claimed
EP-1147107-A1 NOVEL ANGIOGENESIS INHIBITORS Merck & Co., Inc. (US) 2001-10-24 EP claimed
WO-2000043393-A1 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO., INC. (US) 2000-07-27 WO claimed
EP-1147107-A4 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO INC (US) 2002-05-22 EP disclosed
EP-1147107-A1 NOVEL ANGIOGENESIS INHIBITORS Merck & Co., Inc. (US) 2001-10-24 EP disclosed
WO-2000043393-A1 NOVEL ANGIOGENESIS INHIBITORS MERCK & CO., INC. (US) 2000-07-27 WO disclosed