SCHEMBL7558828

SCHEMBL7558828

COC(=O)C#CC#CSc1cc2c(cc1C)C(C)(C)CCC2(C)C

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RXRA P19793 18/20 0.43
RXRG P48443 13/20 0.43
RXRB P28702 12/20 0.43
CYP3A4 P08684 1/20 0.36
RARB P10826 4/20 0.36
RARG P13631 4/20 0.36
RARA P10276 4/20 0.36
HDAC3 O15379 1/20 0.35
HDAC4 P56524 1/20 0.35
HDAC1 Q13547 1/20 0.35
HDAC7 Q8WUI4 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC10 Q969S8 1/20 0.35
HDAC11 Q96DB2 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
HDAC9 Q9UKV0 1/20 0.35
HDAC5 Q9UQL6 1/20 0.35
CYP26A1 O43174 2/20 0.34
PPARG P37231 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7560408 0.86 RXRA (0.49) RXRARXRGRXRBCYP3A4RARB
SCHEMBL6472984 0.76 CYP26A1 (0.46) RXRARXRGRXRBRARBRARG
SCHEMBL6473142 0.75 RXRA (0.36) RXRARXRGRXRBCYP3A4RARB
SCHEMBL7573999 0.73 RXRA (0.41) RXRARXRGRXRBCYP3A4RARB
SCHEMBL7558937 0.72 RXRA (0.48) RXRARXRGRXRBRARBRARG
SCHEMBL7558942 0.72 RXRA (0.48) RXRARXRGRXRBRARBRARG
SCHEMBL7562932 0.71 RXRA (0.40) RXRARXRGRXRBRARBRARG
SCHEMBL7562936 0.71 RXRA (0.40) RXRARXRGRXRBRARBRARG
SCHEMBL7559396 0.70 RXRA (0.47) RXRARXRGRXRBRARBRARG
SCHEMBL8014334 0.66 RXRA (0.60) RXRARXRGRXRBCYP3A4RARB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0986537-B1 NOVEL HETEROETHYNYLENE COMPOUNDS AND PHARMACEUTICAL AND COSMETIC COMPOSITIONS CONTAINING SAME GALDERMA RES & DEV (FR) 2002-08-07 EP claimed