SCHEMBL7559638

SCHEMBL7559638

O=C1C=C(Nc2cccc(C(F)(F)F)c2)CS1

nearest known ligand 0.53

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 10/20 0.53
THRB P10828 1/20 0.47
ADORA2A P29274 1/20 0.46
IDH2 P48735 2/20 0.46
DHODH Q02127 1/20 0.45
ALDH1A1 P00352 2/20 0.44
RAPGEF4 Q8WZA2 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7527253 0.83 MAPT (0.60) ALDH1A1MEN1KMT2AGAAMAPT
SCHEMBL7557829 0.82 KMT2A (0.43) KIF11DHODHMEN1KMT2AMAPT
SCHEMBL15913218 0.77 KIF11 (0.53) KIF11ADORA2AIDH2DHODHALDH1A1
SCHEMBL7520161 0.74 KIF11 (0.52) KIF11ADORA2AIDH2DHODHALDH1A1
SCHEMBL7528061 0.74 KIF11 (0.52) KIF11ADORA2AIDH2DHODHRAPGEF4
SCHEMBL15992074 0.74 KIF11 (0.52) KIF11ADORA2AIDH2DHODHALDH1A1
SCHEMBL394991 0.74 KIF11 (0.70) KIF11THRBADORA2AIDH2ALDH1A1
SCHEMBL15913806 0.72 ALDH1A1 (0.47) KIF11ADORA2AIDH2DHODHALDH1A1
SCHEMBL17477726 0.72 KIF11 (0.50) KIF11ADORA2AIDH2DHODHALDH1A1
SCHEMBL19409877 0.72 IDH2 (0.53) KIF11ADORA2AIDH2DHODHALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173420-A2 HETEROCYCLIC COMPOUNDS HAVING ANTITUMOR ACTIVITY Novuspharma S.p.A. (IT) 2002-01-23 EP disclosed
WO-2000053581-A2 HETEROCYCLIC COMPOUNDS HAVING ANTITUMOR ACTIVITY NOVUSPHARMA S.P.A. (IT) 2000-09-14 WO disclosed