SCHEMBL7528061

SCHEMBL7528061

O=C1C=C(Nc2cccc(C(F)(F)F)c2)CN1

nearest known ligand 0.52

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 11/20 0.52
AKR1C3 P42330 2/20 0.49
AKR1C2 P52895 2/20 0.49
HTT P42858 1/20 0.46
ADORA2A P29274 1/20 0.46
IDH2 P48735 2/20 0.46
RXFP1 Q9HBX9 1/20 0.45
DHODH Q02127 1/20 0.45
RAPGEF4 Q8WZA2 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17477726 0.86 KIF11 (0.50) KIF11AKR1C3AKR1C2HTTADORA2A
SCHEMBL7524850 0.79 IDO1 (0.47) RAPGEF4
SCHEMBL17477740 0.78 KIF11 (0.47) KIF11AKR1C3AKR1C2HTTIDH2
SCHEMBL15913218 0.77 KIF11 (0.53) KIF11AKR1C3AKR1C2ADORA2AIDH2
SCHEMBL7519427 0.75 GRM4 (0.44) RAPGEF4
SCHEMBL7559638 0.74 KIF11 (0.53) KIF11ADORA2AIDH2DHODHRAPGEF4
SCHEMBL15992074 0.74 KIF11 (0.52) KIF11ADORA2AIDH2DHODHRAPGEF4
SCHEMBL7520161 0.74 KIF11 (0.52) KIF11AKR1C3AKR1C2HTTADORA2A
SCHEMBL394991 0.74 KIF11 (0.70) KIF11AKR1C3AKR1C2HTTADORA2A
SCHEMBL15913806 0.72 ALDH1A1 (0.47) KIF11HTTADORA2AIDH2RXFP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1173420-A2 HETEROCYCLIC COMPOUNDS HAVING ANTITUMOR ACTIVITY Novuspharma S.p.A. (IT) 2002-01-23 EP disclosed
WO-2000053581-A2 HETEROCYCLIC COMPOUNDS HAVING ANTITUMOR ACTIVITY NOVUSPHARMA S.P.A. (IT) 2000-09-14 WO disclosed