SCHEMBL7562999

SCHEMBL7562999

COC(=O)c1c(OS(C)(=O)=O)ccc2cc(C(=N)N)ccc12

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PLAU P00749 16/20 0.46
FTO Q9C0B1 1/20 0.44
PLG P00747 7/20 0.43
F2 P00734 7/20 0.43
PRSS1 P07477 7/20 0.43
KLK1 P06870 4/20 0.43
LCK P06239 1/20 0.41
NCEH1 Q6PIU2 1/20 0.41
KLKB1 P03952 5/20 0.39
PLAT P00750 4/20 0.39
C1R P00736 1/20 0.38
F10 P00742 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7563375 0.88 PLAU (0.43) PLAUFTOPLGF2PRSS1
SCHEMBL7562995 0.83 LCK (0.52) PLAUFTOPLGF2PRSS1
SCHEMBL7563090 0.81 FTO (0.48) PLAUFTOPLGF2PRSS1
SCHEMBL7564853 0.81 PLAU (0.43) PLAUFTOPLGF2PRSS1
SCHEMBL7562843 0.80 LCK (0.57) PLAUFTOPLGF2PRSS1
SCHEMBL7326867 0.80 KDM4E (0.43) PLAUFTOPLGF2PRSS1
SCHEMBL7564461 0.78 PLAU (0.42) PLAUFTOPLGF2PRSS1
SCHEMBL7332586 0.74 PRSS1 (0.59) PLAUPLGF2PRSS1KLK1
SCHEMBL15902277 0.73 PLAU (0.65) PLAUFTOPLGF2PRSS1
SCHEMBL7563372 0.73 PLAU (0.47) PLAUFTOPLGF2PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802179-B1 SUBSTITUTED AMIDINONAPHTHYL ESTER DERIVATIVES TORII PHARMACEUTICAL CO LTD (JP) 2002-08-21 EP disclosed
US-5885990-A FIBRINOLYSIS PROMOTING ACTION; THROMBOLYSIS ACTION TORII PHARMACEUTICAL CO., LTD. (JP) 1999-03-23 US disclosed
EP-0802179-A1 SUBSTITUTED AMIDINONAPHTHYL ESTER DERIVATIVES TORII PHARMACEUTICAL CO., LTD. (JP) 1997-10-22 EP disclosed