SCHEMBL7563375

SCHEMBL7563375

CS(=O)(=O)Oc1ccc2cc(C(=N)N)ccc2c1C(=O)O

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PLAU P00749 18/20 0.43
PLG P00747 7/20 0.43
KLK1 P06870 5/20 0.43
F2 P00734 5/20 0.43
PRSS1 P07477 5/20 0.43
FTO Q9C0B1 1/20 0.41
PLAT P00750 4/20 0.39
KLKB1 P03952 3/20 0.39
F12 P00748 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7562999 0.88 PLAU (0.46) PLAUPLGKLK1F2PRSS1
SCHEMBL7564461 0.82 PLAU (0.42) PLAUPLGKLK1F2PRSS1
SCHEMBL7563372 0.80 PLAU (0.47) PLAUPLGKLK1F2PRSS1
SCHEMBL7332931 0.79 PLAU (0.40) PLAUPLGKLK1F2PRSS1
SCHEMBL16510334 0.78 METAP2 (0.48)
SCHEMBL30525132 0.78 METAP2 (0.48)
SCHEMBL7563955 0.78 FTO (0.48) PLAUPLGKLK1F2PRSS1
SCHEMBL7564853 0.78 PLAU (0.43) PLAUPLGKLK1F2PRSS1
SCHEMBL29769933 0.74 NCEH1 (0.40) PLAUPLGKLK1F2PRSS1
SCHEMBL31266874 0.74 FTO (0.54) PLAUPLGKLK1F2PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802179-B1 SUBSTITUTED AMIDINONAPHTHYL ESTER DERIVATIVES TORII PHARMACEUTICAL CO LTD (JP) 2002-08-21 EP disclosed
US-5885990-A FIBRINOLYSIS PROMOTING ACTION; THROMBOLYSIS ACTION TORII PHARMACEUTICAL CO., LTD. (JP) 1999-03-23 US disclosed
EP-0802179-A1 SUBSTITUTED AMIDINONAPHTHYL ESTER DERIVATIVES TORII PHARMACEUTICAL CO., LTD. (JP) 1997-10-22 EP disclosed