Bromide

Bromide

SCHEMBL7564429

Br.Nc1cc(CBr)nc(N)n1

nearest known ligand 0.52

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.35
MEN1 O00255 1/20 0.35
NPC1 O15118 1/20 0.35
PABPC1 P11940 1/20 0.35
RAB9A P51151 1/20 0.35
KMT2A Q03164 1/20 0.35
NOS3 P29474 3/20 0.33
NOS2 P35228 3/20 0.33
TDP1 Q9NUW8 1/20 0.33
CCR1 P32246 1/20 0.33
HRH4 Q9H3N8 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
HSP90AB1 P08238 1/20 0.32
DYRK1A Q13627 1/20 0.32
NOS1 P29475 2/20 0.31
CYP3A4 P08684 1/20 0.31
BLM P54132 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7563064 0.98 MAPT (0.36) MAPTMEN1NPC1PABPC1RAB9A
Bromide SCHEMBL27537591 0.83 NOS2 (0.37) MAPTMEN1NPC1PABPC1RAB9A
SCHEMBL27537579 0.78 NOS2 (0.37) MAPTMEN1NPC1PABPC1RAB9A
SCHEMBL2879873 0.77 CCR1 (0.33) CCR1HSP90AB1
Bromide SCHEMBL27537590 0.77 NOS2 (0.36) MAPTMEN1NPC1PABPC1RAB9A
SCHEMBL2879516 0.76 HSP90AB1 (0.56) MAPTMEN1KMT2AHRH4HSP90AB1
SCHEMBL656121 0.74 MAPT (0.50) MAPTMEN1NPC1PABPC1RAB9A
SCHEMBL7562734 0.74 MAPT (0.34) MAPTMEN1NPC1PABPC1RAB9A
SCHEMBL9067684 0.74 NOS2 (0.39) MAPTNOS3NOS2TDP1CCR1
SCHEMBL6361284 0.74 NOS2 (0.59) NOS3NOS2HRH4HRH3NOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077981-B1 NOVEL CEPHALOSPORIN COMPOUNDS, PROCESSES FOR PREPARATION THEREOF AND ANTIMICROBIAL COMPOSITIONS CONTAINING THE SAME LG CHEMICAL LTD (KR) 2002-08-07 EP disclosed
EP-1077981-A1 NOVEL CEPHALOSPORIN COMPOUNDS, PROCESSES FOR PREPARATION THEREOF AND ANTIMICROBIAL COMPOSITIONS CONTAINING THE SAME LG CHEMICAL LIMITED (KR) 2001-02-28 EP disclosed
WO-1999058535-A1 NOVEL CEPHALOSPORIN COMPOUNDS, PROCESSES FOR PREPARATION THEREOF AND ANTIMICROBIAL COMPOSITIONS CONTAINING THE SAME LG CHEMICAL LTD. (KR) 1999-11-18 WO disclosed