SCHEMBL9067684

SCHEMBL9067684

Nc1cc(N)nc(CBr)c1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 10/20 0.39
NOS3 P29474 6/20 0.39
NOS1 P29475 6/20 0.36
MAPT P10636 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CCR1 P32246 1/20 0.34
CYP3A4 P08684 1/20 0.32
BLM P54132 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13688177 0.76 MAPT (0.50) NOS2NOS3NOS1MAPTTDP1
SCHEMBL7563064 0.76 MAPT (0.36) NOS2NOS3NOS1MAPTTDP1
SCHEMBL10399435 0.76 NOS2 (0.65) NOS2NOS3NOS1
Bromide SCHEMBL7564429 0.74 MAPT (0.35) NOS2NOS3NOS1MAPTTDP1
SCHEMBL2088900 0.74 NOS2 (0.38) NOS2NOS3NOS1
SCHEMBL1317980 0.73
SCHEMBL9007840 0.69 ALDH1A1 (0.47) NOS2NOS3NOS1MAPTTDP1
SCHEMBL2879873 0.65 CCR1 (0.33) CCR1
SCHEMBL2879516 0.64 HSP90AB1 (0.56) MAPT
SCHEMBL9637847 0.64 KCNH2 (0.37) NOS2NOS3CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5536724-A Antiinflammatory and antineoplastic 5-deazaaminopterins and 5,10-dideazaaminopterins SRI INTERNATIONAL (US) 1996-07-16 US disclosed