SCHEMBL7564431

SCHEMBL7564431

CC1=Cc2c(-c3cnc4ccccc4c3)cccc2C1[Si](C)(C)C1C(C)=Cc2c(-c3cnc4ccccc4c3)cccc21

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.42
CREBBP Q92793 2/20 0.42
PDGFRB P09619 4/20 0.40
PDGFRA P16234 4/20 0.40
CYP1A2 P05177 1/20 0.40
BIRC5 O15392 1/20 0.40
MAP4K4 O95819 1/20 0.39
CSNK1G2 P78368 1/20 0.39
CLK4 Q9HAZ1 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
MAP4K5 Q9Y4K4 1/20 0.39
PARP10 Q53GL7 1/20 0.38
PARP11 Q9NR21 1/20 0.38
CYP2A6 P11509 1/20 0.38
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
AKR1C3 P42330 2/20 0.36
AKR1C2 P52895 2/20 0.36
PFKFB3 Q16875 1/20 0.36
NPC1 O15118 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3159292 0.82 GSTP1 (0.38) CYP1A2ALDH1A1
SCHEMBL8675237 0.80 BRD4 (0.39) BRD4CREBBPPDGFRBPDGFRACYP1A2
Hydrochloric Acid SCHEMBL5170143 0.80 GSTP1 (0.36) CYP1A2ALDH1A1
Hydrochloric Acid SCHEMBL7569789 0.79 PARP10 (0.40) BRD4CREBBPPDGFRBPDGFRACYP1A2
Hydrochloric Acid SCHEMBL8675926 0.79 BRD4 (0.38) BRD4CREBBPPDGFRBPDGFRACYP1A2
SCHEMBL8675236 0.79 BRD4 (0.38) BRD4CREBBPPDGFRBPDGFRACYP1A2
SCHEMBL29366427 0.79 PDCD1 (0.34) BRD4CYP2A6NPC1ALDH1A1RAB9A
SCHEMBL61908 0.79 PDCD1 (0.34) BRD4CYP2A6NPC1ALDH1A1RAB9A
SCHEMBL5953421 0.78 PARP10 (0.37) BRD4CREBBPPDGFRBPDGFRACYP1A2
Hydrochloric Acid SCHEMBL7562438 0.77 PARP10 (0.39) BRD4CREBBPPDGFRBPDGFRACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0743317-B1 Metallocenes comprising a heterocycle and catalysts containing them BASELL POLYOLEFINE GMBH (DE) 2002-08-28 EP disclosed
US-5840947-A Organometallic compound TARGOR GMBH (DE) 1998-11-24 US disclosed
EP-0743317-A2 Metallocenes comprising a heterocycle and catalysts containing them HOECHST AKTIENGESELLSCHAFT (DE) 1996-11-20 EP disclosed