SCHEMBL7564651

SCHEMBL7564651

O=C(O)CCCOc1ccc(CO)cc1[N+](=O)[O-]

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.51
MAPT P10636 3/20 0.51
PRSS1 P07477 4/20 0.48
ALPG P10696 1/20 0.47
LMNA P02545 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
KDM4E B2RXH2 2/20 0.46
GAA P10253 1/20 0.46
TTR P02766 1/20 0.46
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
PDCD1 Q15116 1/20 0.45
CD274 Q9NZQ7 1/20 0.45
HTT P42858 1/20 0.44
THRA P10827 1/20 0.44
THRB P10828 1/20 0.44
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11953000 0.83 MAPT (0.70) ALDH1A1MAPTPRSS1ALPGLMNA
SCHEMBL4120809 0.83 PRSS1 (0.50) ALDH1A1MAPTPRSS1LMNAKDM4E
SCHEMBL5968434 0.82 MAPT (0.65) ALDH1A1MAPTPRSS1ALPGLMNA
SCHEMBL2213228 0.80 PRSS1 (0.56) ALDH1A1MAPTPRSS1LMNAKDM4E
SCHEMBL7567675 0.80 ALDH1A1 (0.55) ALDH1A1MAPTPRSS1LMNANPSR1
SCHEMBL12781092 0.80 ALDH1A1 (0.50) ALDH1A1MAPTPRSS1ALPGLMNA
SCHEMBL8164415 0.79 NPC1 (0.70) ALDH1A1MAPTLMNAKDM4EMEN1
SCHEMBL9320548 0.79 NPC1 (0.70) ALDH1A1MAPTLMNAKDM4EMEN1
SCHEMBL5913597 0.79 LMNA (0.62) ALDH1A1MAPTALPGLMNANPSR1
SCHEMBL27837027 0.78 CYSLTR2 (0.55) ALDH1A1MAPTPRSS1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0689845-B1 Conjugates of methyltrithio antitumor agents and intermediates for their synthesis AMERICAN CYANAMID CO (US) 2002-09-04 EP disclosed
US-5877296-A REACTING DISULFIDE ANALOGS OF CALICHEAMICIN FAMILY WITH A CARRIER SUCH AS PROTEIN, PEPTIDE, MONO AND POLYCLONAL ANTIBODIES, THEIR ANTIGEN-RECOGNIZING FRAGMENTS AND CHEMICALLY OR GENETICALLY ENGINEERED COUNTERPARTS AMERICAN CYANAMID COMPANY (US) 1999-03-02 US disclosed
US-5773001-A ANTIGROWTH AGENTS AMERICAN CYANAMID COMPANY (US) 1998-06-30 US disclosed
US-5767285-A USEFUL FOR CONSTRUCTING DRUG CONJUGATES; ANTIBIOTIC ANTITUMOR AGENTS AMERICAN CYANAMID COMPANY (US) 1998-06-16 US disclosed
US-5739116-A DISULFIDE DERIVATIVE OF CALICHEAMICIN FAMILY; ANTITUMOR ANTIBIOTICS AMERICAN CYANAMID COMPANY (US) 1998-04-14 US disclosed
EP-0689845-A2 Conjugates of methyltrithio antitumor agents and intermediates for their synthesis AMERICAN CYANAMID COMPANY (US) 1996-01-03 EP disclosed