SCHEMBL7564915

SCHEMBL7564915

N#Cc1ccccc1N1CCN(C[C@H](O)COc2ccc(-c3onc4cc(F)ccc34)cc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 4/20 0.52
HTR7 P34969 4/20 0.52
HSP90AB1 P08238 2/20 0.51
DRD2 P14416 2/20 0.45
MAPT P10636 3/20 0.45
ALDH1A1 P00352 3/20 0.44
LMNA P02545 2/20 0.44
CACNA1G O43497 2/20 0.44
TP53 P04637 1/20 0.44
GAA P10253 1/20 0.44
MAPK1 P28482 1/20 0.44
HTT P42858 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KCNH2 Q12809 1/20 0.44
KDM4E B2RXH2 2/20 0.43
ABCB1 P08183 2/20 0.43
ADRB3 P13945 1/20 0.43
HPGD P15428 1/20 0.42
HSD17B10 Q99714 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7564923 1.00 HTR1A (0.52) HTR1AHTR7HSP90AB1DRD2MAPT
SCHEMBL1383563 0.87 MAPT (0.55) HTR7MAPTALDH1A1LMNACACNA1G
SCHEMBL1383560 0.87 MAPT (0.55) HTR7MAPTALDH1A1LMNACACNA1G
SCHEMBL5370498 0.86 HTR1A (0.53) HTR1AHTR7HSP90AB1DRD2MAPT
SCHEMBL5363235 0.86 HTR1A (0.53) HTR1AHTR7HSP90AB1DRD2MAPT
SCHEMBL5363239 0.86 HTR1A (0.53) HTR1AHTR7HSP90AB1DRD2MAPT
SCHEMBL7569775 0.85 HTR1A (0.53) HTR1AHTR7HSP90AB1MAPTALDH1A1
SCHEMBL7492035 0.85 MAPT (0.54) MAPTALDH1A1LMNATP53GAA
SCHEMBL7492021 0.85 MAPT (0.54) MAPTALDH1A1LMNATP53GAA
SCHEMBL7493514 0.85 MAPT (0.54) MAPTALDH1A1LMNATP53GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216244-A1 Benzisoxazolyl-, pyridoisoxazolyl- and benzthienyl-phenoxy derivatives useful as D4 antagonists Aventis Pharmaceuticals Inc. (US) 2002-06-26 EP disclosed
WO-2001019821-A1 BENZISOXAZOLYL-, PYRIDOISOXAZOLYL- AND BENZTHIENYL-PHENOXY DERIVATIVES USEFUL AS D4 ANTAGONISTS AVENTIS PHARMACEUTICALS INC. (US) 2001-03-22 WO disclosed