SCHEMBL7569775

SCHEMBL7569775

N#Cc1ccccc1N1CCN(CC(O)COc2ccc(-c3occ4cc(F)ccc34)cc2)CC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 2/20 0.53
HTR7 P34969 2/20 0.53
HSP90AB1 P08238 2/20 0.52
MAPT P10636 3/20 0.47
ALDH1A1 P00352 5/20 0.45
LMNA P02545 2/20 0.45
CACNA1G O43497 2/20 0.45
TP53 P04637 1/20 0.45
GAA P10253 1/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
KCNH2 Q12809 1/20 0.45
KDM4E B2RXH2 3/20 0.44
ABCB1 P08183 2/20 0.43
HSD17B10 Q99714 2/20 0.43
HPGD P15428 1/20 0.43
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
USP2 O75604 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7564923 0.85 HTR1A (0.52) HTR1AHTR7HSP90AB1MAPTALDH1A1
SCHEMBL7564915 0.85 HTR1A (0.52) HTR1AHTR7HSP90AB1MAPTALDH1A1
SCHEMBL7565949 0.84 KDM4E (0.51) HTR1AMAPTALDH1A1LMNACACNA1G
SCHEMBL7572390 0.83 KDM4E (0.58) MAPTALDH1A1LMNACACNA1GHTT
SCHEMBL1382258 0.83 ATM (0.56) SMN1; SMN2KDM4EABCB1HSD17B10KMT2A
SCHEMBL5370498 0.82 HTR1A (0.53) HTR1AHTR7HSP90AB1MAPTALDH1A1
SCHEMBL5363235 0.82 HTR1A (0.53) HTR1AHTR7HSP90AB1MAPTALDH1A1
SCHEMBL5363239 0.82 HTR1A (0.53) HTR1AHTR7HSP90AB1MAPTALDH1A1
SCHEMBL7572169 0.82 PKM (0.57) ALDH1A1LMNAGAAMAPK1SMN1; SMN2
SCHEMBL7564076 0.82 PKM (0.43) HTR1AMAPTALDH1A1CACNA1GKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1216244-A1 Benzisoxazolyl-, pyridoisoxazolyl- and benzthienyl-phenoxy derivatives useful as D4 antagonists Aventis Pharmaceuticals Inc. (US) 2002-06-26 EP disclosed
WO-2001019821-A1 BENZISOXAZOLYL-, PYRIDOISOXAZOLYL- AND BENZTHIENYL-PHENOXY DERIVATIVES USEFUL AS D4 ANTAGONISTS AVENTIS PHARMACEUTICALS INC. (US) 2001-03-22 WO disclosed