SCHEMBL7564976

SCHEMBL7564976

O=[N+]([O-])c1cccc(-c2nc(CS(=O)(=O)CCO)no2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.61
NPC1 O15118 7/20 0.55
RAB9A P51151 7/20 0.55
MAPT P10636 6/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2C9 P11712 1/20 0.52
CYP2C19 P33261 1/20 0.52
CHRNB2 P17787 1/20 0.50
CHRNA5 P30532 1/20 0.50
CHRNA4 P43681 1/20 0.50
GRM5 P41594 1/20 0.49
MAPK1 P28482 1/20 0.45
SMN1; SMN2 Q16637 3/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
CA13 Q8N1Q1 1/20 0.43
PSMB8 P28062 1/20 0.41
MEN1 O00255 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8399931 0.86 NPC1 (0.48) ALDH1A1NPC1RAB9AMAPTCHRNB2
SCHEMBL7569714 0.81 ALDH1A1 (0.45) ALDH1A1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL7566184 0.81 ALDH1A1 (0.63) ALDH1A1NPC1RAB9AMAPTCYP1A2
SCHEMBL22347443 0.78 ALDH1A1 (0.81) ALDH1A1NPC1RAB9AMAPTCYP1A2
SCHEMBL1544191 0.78 ALDH1A1 (0.73) ALDH1A1NPC1RAB9AMAPTCYP1A2
SCHEMBL11370147 0.74 ALDH1A1 (0.86) ALDH1A1NPC1RAB9AMAPTCYP1A2
SCHEMBL8404853 0.73 MEN1 (0.47) ALDH1A1NPC1RAB9AMAPTSMN1; SMN2
SCHEMBL3016134 0.73 TSHR (0.53) ALDH1A1CYP1A2CYP3A4CYP2C9CYP2C19
SCHEMBL12653007 0.72 NPC1 (0.70) ALDH1A1NPC1RAB9AMAPTCYP1A2
SCHEMBL10867150 0.69 ALDH1A1 (0.55) ALDH1A1NPC1RAB9AMAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0929610-B1 REACTIVE DYES WITH A HETEROCYCLIC ANCHOR DYSTAR TEXTILFARBEN GMBH & CO (DE) 2002-08-28 EP disclosed
US-6197941-B1 TRIAZINE, METALLIZED, AZO, ANTHRAQUINONE, FORMAZAN, PHTHALOCYANINE, AND DIOXAZINE DYES BASF AKTIENGESELLSCHAFT (DE) 2001-03-06 US disclosed
EP-0842163-B1 BENZENE DERIVATIVES WITH A HETEROCYCLIC GROUP BASF AG (DE) 1999-11-03 EP disclosed
US-5886187-A Benzene derivatives having a heterocyclic radical BASF AKTIENGESELLSCHAFT (DE) 1999-03-23 US disclosed
EP-0842163-A1 BENZENE DERIVATIVES WITH A HETEROCYCLIC GROUP BASF AKTIENGESELLSCHAFT (DE) 1998-05-20 EP disclosed
WO-1997005124-A1 BENZENE DERIVATIVES WITH A HETEROCYCLIC GROUP BASF AKTIENGESELLSCHAFT (DE) 1997-02-13 WO disclosed