SCHEMBL7565031

SCHEMBL7565031

CN(C)C(=O)C1Cc2c(N)cccc2NC1=O.CN(C)C(=O)C1Cc2c(NC(=O)OCc3ccccc3)cccc2NC1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.43
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42
IDO1 P14902 4/20 0.39
TDO2 P48775 2/20 0.39
CYP3A4 P08684 2/20 0.38
TSHR P16473 1/20 0.38
BRD4 O60885 1/20 0.38
CREBBP Q92793 1/20 0.38
PARP1 P09874 1/20 0.38
HDAC3 O15379 2/20 0.38
HDAC1 Q13547 2/20 0.38
HDAC2 Q92769 2/20 0.38
PLAU P00749 1/20 0.37
PTPN1 P18031 1/20 0.37
PDE3B Q13370 1/20 0.36
PDE3A Q14432 1/20 0.36
MAOB P27338 3/20 0.36
KDM1A O60341 2/20 0.36
MAOA P21397 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7480378 0.95 CASP3 (0.47) CASP3NPC1RAB9AIDO1TDO2
SCHEMBL7484149 0.81 DDB1 (0.33) BRD4CREBBPPARP1
SCHEMBL7833079 0.75 TSHR (0.45) NPC1RAB9ACYP3A4TSHRPTPN1
SCHEMBL3811403 0.69 NPC1 (0.68) CASP3NPC1RAB9ACYP3A4HDAC3
SCHEMBL3784499 0.66 NPC1 (0.59) CASP3NPC1RAB9AHDAC3HDAC1
SCHEMBL3789479 0.65 CASP3 (0.60) CASP3NPC1RAB9AHDAC3HDAC1
SCHEMBL3789191 0.65 NPC1 (0.61) CASP3NPC1RAB9AHDAC3HDAC1
SCHEMBL7836971 0.65 CREBBP (0.46) NPC1BRD4CREBBP
SCHEMBL3792921 0.65 NPC1 (0.57) CASP3NPC1RAB9AHDAC3HDAC1
SCHEMBL1961986 0.64 NPC1 (0.50) CASP3NPC1RAB9ATSHRPLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227090-A1 AMINE DERIVATIVES Tadeka Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed