SCHEMBL7480378

SCHEMBL7480378

CN(C)C(=O)C1Cc2c(NC(=O)OCc3ccccc3)cccc2NC1=O

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 1/20 0.47
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
IDO1 P14902 4/20 0.43
TDO2 P48775 2/20 0.43
CYP3A4 P08684 2/20 0.42
TSHR P16473 1/20 0.42
BRD4 O60885 1/20 0.41
CREBBP Q92793 1/20 0.41
PARP1 P09874 1/20 0.41
PTPN1 P18031 1/20 0.40
PDE3B Q13370 1/20 0.39
PDE3A Q14432 1/20 0.39
MAOB P27338 2/20 0.39
CCKBR P32239 1/20 0.38
PLAU P00749 1/20 0.38
MGLL Q99685 1/20 0.38
KDM1A O60341 1/20 0.37
MAOA P21397 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7565031 0.95 CASP3 (0.43) CASP3NPC1RAB9AIDO1TDO2
SCHEMBL7833079 0.80 TSHR (0.45) NPC1RAB9ACYP3A4TSHRPTPN1
SCHEMBL7484149 0.71 DDB1 (0.33) BRD4CREBBPPARP1
SCHEMBL7836971 0.68 CREBBP (0.46) NPC1BRD4CREBBP
SCHEMBL7945076 0.67 NPC1 (0.49) NPC1RAB9ATSHRPTPN1PDE3B
SCHEMBL30522295 0.67 NPC1 (0.69) CASP3NPC1RAB9APTPN1MAOB
SCHEMBL16193532 0.67 NPC1 (0.69) CASP3NPC1RAB9APTPN1MAOB
SCHEMBL2233522 0.67 NPC1 (0.69) CASP3NPC1RAB9APTPN1MAOB
SCHEMBL472400 0.66 TRPV1 (0.53) CASP3NPC1RAB9APTPN1PLAU
SCHEMBL10874779 0.66 NPC1 (0.68) NPC1RAB9ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1227090-A1 AMINE DERIVATIVES Tadeka Chemical Industries, Ltd. (JP) 2002-07-31 EP disclosed