SCHEMBL7565046

SCHEMBL7565046

CC(C)c1[c]c(-c2ccc(F)cc2)cc(C(C)C)n1

nearest known ligand 0.37

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.37
HTR2C P28335 2/20 0.37
HTR2B P41595 2/20 0.37
GCGR P47871 11/20 0.33
PTGS1 P23219 1/20 0.32
PTGS2 P35354 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2C19 P33261 1/20 0.31
SCN9A Q15858 1/20 0.31
MAPK14 Q16539 2/20 0.30
MAPK13 O15264 1/20 0.30
MAPK12 P53778 1/20 0.30
MAPK11 Q15759 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8846284 0.79 MAPT (0.43) CYP1A2CYP2C19
SCHEMBL6013166 0.69 SCN9A (0.39) HTR2AHTR2CHTR2BGCGRSCN9A
SCHEMBL8201704 0.68 ADORA2A (0.43) GCGRSCN9AMAPK14
SCHEMBL12202948 0.67 ADORA3 (0.41) HTR2BGCGR
SCHEMBL12228276 0.67 KDM4E (0.45) HTR2BSCN9A
SCHEMBL3840856 0.66 AURKA (0.56) HTR2BPTGS2CYP1A2MAPK14
SCHEMBL28094104 0.66 NOS3 (0.44) HTR2BCYP1A2CYP2C19SCN9A
SCHEMBL2337367 0.66 ADORA3 (0.43) GCGRSCN9A
SCHEMBL9302391 0.65 APP (0.42)
SCHEMBL9302519 0.65 ADORA2A (0.43) SCN9AMAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705837-B1 Preparation of 3-Oxy-5-oxo-6-heptenoic acid derivatives UBE INDUSTRIES (JP) 2002-08-07 EP disclosed
US-5744604-A Preparation of 3-oxy-5-oxo-6-heptenoic acid derivatives UBE INDUSTRIES, LTD. (JP) 1998-04-28 US disclosed
US-5677455-A Preparation of 3-oxy-5-oxo-6-heptenoic acid derivatives UBE INDUSTRIES, LTD. (JP) 1997-10-14 US disclosed
EP-0705837-A2 Preparation of 3-Oxy-5-oxo-6-heptenoic acid derivatives UBE INDUSTRIES, LTD. (JP) 1996-04-10 EP disclosed