SCHEMBL7567330

SCHEMBL7567330

Nc1cc(COC(=O)Nc2cc(F)cc(F)c2)cc(Nc2c3ccccc3nc3ccccc23)c1

nearest known ligand 0.73

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TOP2A P11388 9/20 0.73
TOP2B Q02880 8/20 0.73
KDM4E B2RXH2 2/20 0.44
POLB P06746 2/20 0.44
GLA P06280 1/20 0.44
KDM1A O60341 2/20 0.43
HDAC3 O15379 3/20 0.42
HDAC4 P56524 3/20 0.42
HDAC1 Q13547 3/20 0.42
HDAC7 Q8WUI4 3/20 0.42
HDAC2 Q92769 3/20 0.42
HDAC8 Q9BY41 3/20 0.42
HDAC6 Q9UBN7 3/20 0.42
HDAC9 Q9UKV0 3/20 0.42
HDAC5 Q9UQL6 3/20 0.42
ACHE P22303 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
MITF O75030 1/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7561269 0.93 TOP2A (0.66) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL7564074 0.93 TOP2A (0.66) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL7561273 0.92 TOP2A (0.70) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL7568574 0.92 TOP2A (0.73) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL3981533 0.91 TOP2A (0.80) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL7563689 0.89 TOP2A (0.77) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL7564525 0.89 TOP2A (0.61) TOP2ATOP2BPOLBKDM1ARAD52
SCHEMBL7569259 0.89 TOP2A (0.61) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL7563590 0.88 TOP2A (0.70) TOP2ATOP2BKDM4EPOLBGLA
SCHEMBL7567582 0.88 TOP2A (0.73) TOP2ATOP2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20020111491-A1 9-aminoacridine derivatives and process for the preparation thereof SAMJIN PHARMACEUTICAL CO., LTD. (KR) 2002-08-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020111491-A1 9-aminoacridine derivatives and process for the preparation thereof ALKBH1, ADCY9, CCR9 TOP2A 1105/4885TOP2B 841/4885KDM4E 1567/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.