SCHEMBL7567397

SCHEMBL7567397

CNCCCNC(=O)c1cccc2cc3cccc(C(F)(F)F)c3nc12

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 3/20 0.47
HDAC6 Q9UBN7 2/20 0.47
AOX1 Q06278 1/20 0.46
TP53 P04637 1/20 0.41
PARP1 P09874 1/20 0.40
HDAC3 O15379 2/20 0.40
TP53BP1 Q12888 1/20 0.40
GPR52 Q9Y2T5 1/20 0.39
RAD52 P43351 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39
TSHR P16473 1/20 0.39
HTT P42858 1/20 0.39
PTGES O14684 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7566458 0.86 AOX1 (0.52) HDAC1HDAC6AOX1TP53RAD52
SCHEMBL7107762 0.84 AOX1 (0.65) HDAC1HDAC6AOX1PARP1RAD52
SCHEMBL7573617 0.83 HDAC1 (0.49) HDAC1HDAC6AOX1RAD52TSHR
SCHEMBL8624357 0.83 HDAC1 (0.49) HDAC1HDAC6AOX1RAD52TSHR
SCHEMBL8413595 0.81 AOX1 (0.54) HDAC1HDAC6AOX1HDAC3RAD52
SCHEMBL8412027 0.81 AOX1 (0.48) HDAC1HDAC6AOX1TP53BP1RAD52
SCHEMBL8415169 0.81 HDAC1 (0.47) HDAC1HDAC6AOX1TP53RAD52
SCHEMBL7570699 0.79 HDAC1 (0.45) HDAC1HDAC6AOX1RAD52TSHR
SCHEMBL7572168 0.77 AOX1 (0.57) HDAC1HDAC6AOX1RAD52MEN1
SCHEMBL7570661 0.77 AOX1 (0.57) HDAC1HDAC6AOX1TP53BP1RAD52

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0934278-B1 BIS(ACRIDINECARBOXAMIDE) AND BIS(PHENAZINECARBOXAMIDE) AS ANTITUMOUR AGENTS XENOVA LTD (GB) 2002-09-04 EP claimed